SCHEMBL8060040

SCHEMBL8060040

COCC1CCCN1c1cc2nc(S)[nH]c2cc1F

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 6/20 0.39
ROCK2 O75116 1/20 0.39
ROCK1 Q13464 1/20 0.39
CDC42BPB Q9Y5S2 1/20 0.39
ADORA2A P29274 6/20 0.37
ADORA1 P30542 4/20 0.37
MAP4K1 Q92918 1/20 0.36
CRHR1 P34998 1/20 0.36
NMT1 P30419 2/20 0.36
CASP7 P55210 1/20 0.34
PDE10A Q9Y233 1/20 0.34
CYP1A2 P05177 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADORA2B P29275 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8106931 0.75 OPRL1 (0.45) OPRL1ROCK2ROCK1CDC42BPBMAP4K1
SCHEMBL8059824 0.74 OPRL1 (0.44) OPRL1ROCK2ROCK1CDC42BPBMAP4K1
SCHEMBL8075644 0.74 ADORA2A (0.43) ROCK2ROCK1CDC42BPBADORA2AADORA1
SCHEMBL8071108 0.73 MAP4K1 (0.39) ROCK2ROCK1CDC42BPBADORA2AADORA1
SCHEMBL8071080 0.71 EGLN1 (0.52) OPRL1
SCHEMBL8070777 0.71 EGLN1 (0.52) OPRL1
SCHEMBL8069366 0.70 OPRL1 (0.66) OPRL1
SCHEMBL8074378 0.69 OPRL1 (0.46) OPRL1
SCHEMBL2935652 0.69 CHRNB4 (0.43) ROCK2ROCK1CDC42BPBADORA2AADORA1
SCHEMBL8069092 0.69 OPRL1 (0.57) OPRL1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6051570-A ANTIULCER AGENTS DR. REDDY'S RESEARCH FOUNDATION (IN) 2000-04-18 US disclosed
EP-0983263-A1 NOVEL BENZIMIDAZOLE DERIVATIVES AS ANTIULCER AGENTS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 2000-03-08 EP disclosed
WO-1998054172-A1 NOVEL BENZIMIDAZOLE DERIVATIVES AS ANTIULCER AGENTS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 1998-12-03 WO disclosed