SCHEMBL8106931

SCHEMBL8106931

COCc1ccnc(CSc2nc3cc(N4CCCC4COC)c(F)cc3[nH]2)c1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 13/20 0.45
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
CDC42BPB Q9Y5S2 1/20 0.40
NOS2 P35228 3/20 0.39
NOS3 P29474 2/20 0.39
NOS1 P29475 2/20 0.39
CYP1A2 P05177 2/20 0.37
CYP2E1 P05181 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2C8 P10632 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2B6 P20813 2/20 0.37
CYP2C19 P33261 2/20 0.37
MAP4K1 Q92918 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8059824 0.83 OPRL1 (0.44) OPRL1ROCK2ROCK1CDC42BPBCYP1A2
SCHEMBL8060040 0.75 OPRL1 (0.39) OPRL1ROCK2ROCK1CDC42BPBCYP1A2
SCHEMBL8071108 0.69 MAP4K1 (0.39) ROCK2ROCK1CDC42BPBMAP4K1
SCHEMBL8071180 0.67 NOS2 (0.58) OPRL1NOS2NOS3NOS1CYP1A2
SCHEMBL8073907 0.66 OPRL1 (0.37) OPRL1
SCHEMBL8072215 0.65 OPRL1 (0.54) OPRL1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8071079 0.65 OPRL1 (0.58) OPRL1CYP1A2CYP2E1CYP3A4CYP2C8
SCHEMBL8060096 0.65 OPRL1 (0.53) OPRL1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8075357 0.65 OPRL1 (0.53) OPRL1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8070520 0.64 OPRL1 (0.50) OPRL1CYP1A2CYP2E1CYP3A4CYP2C8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0983263-A1 NOVEL BENZIMIDAZOLE DERIVATIVES AS ANTIULCER AGENTS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 2000-03-08 EP disclosed
WO-1998054172-A1 NOVEL BENZIMIDAZOLE DERIVATIVES AS ANTIULCER AGENTS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 1998-12-03 WO disclosed