SCHEMBL8075644

SCHEMBL8075644

COCC1CCCN1c1cc(N)c(N)cc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.43
ADORA1 P30542 4/20 0.43
ROCK2 O75116 1/20 0.41
ROCK1 Q13464 1/20 0.41
CDC42BPB Q9Y5S2 1/20 0.41
CASP7 P55210 3/20 0.38
MAP4K1 Q92918 1/20 0.37
CRHR1 P34998 1/20 0.37
NR1I2 O75469 1/20 0.36
SMARCA2 P51531 1/20 0.36
SMARCA4 P51532 1/20 0.36
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36
PBRM1 Q86U86 1/20 0.36
FFAR2 O15552 1/20 0.35
DRD2 P14416 1/20 0.35
DRD3 P35462 1/20 0.35
KCNH2 Q12809 1/20 0.35
CYP1A2 P05177 1/20 0.35
ADORA3 P0DMS8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8075591 0.84 MAPT (0.48) ADORA2AADORA1CYP1A2
SCHEMBL2935652 0.78 CHRNB4 (0.43) ADORA2AADORA1ROCK2ROCK1CDC42BPB
SCHEMBL8075647 0.76 ADORA2A (0.39) ADORA2AADORA1ROCK2ROCK1CDC42BPB
SCHEMBL8060040 0.74 OPRL1 (0.39) ADORA2AADORA1ROCK2ROCK1CDC42BPB
SCHEMBL13538960 0.73 ROCK2 (0.40) ADORA2AADORA1ROCK2ROCK1CDC42BPB
SCHEMBL9899670 0.72 MAPT (0.54) ADORA2AADORA1ROCK2ROCK1CDC42BPB
SCHEMBL9899672 0.72 MAPT (0.54) ADORA2AADORA1ROCK2ROCK1CDC42BPB
SCHEMBL13638851 0.71 ADORA2A (0.45) ADORA2AADORA1ROCK2ROCK1CDC42BPB
SCHEMBL2447116 0.71 FPR1 (0.47) ADORA2AADORA1ROCK2ROCK1CDC42BPB
SCHEMBL2448887 0.71 FPR1 (0.47) ADORA2AADORA1ROCK2ROCK1CDC42BPB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6051570-A ANTIULCER AGENTS DR. REDDY'S RESEARCH FOUNDATION (IN) 2000-04-18 US disclosed
EP-0983263-A1 NOVEL BENZIMIDAZOLE DERIVATIVES AS ANTIULCER AGENTS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 2000-03-08 EP disclosed
WO-1998054172-A1 NOVEL BENZIMIDAZOLE DERIVATIVES AS ANTIULCER AGENTS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 1998-12-03 WO disclosed