SCHEMBL8060646

SCHEMBL8060646

CCc1cc2c(cc1C(=O)OC)S(=O)(=O)CC(C)(C)N2C

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.35
KDM4E B2RXH2 6/20 0.35
MAPT P10636 2/20 0.35
HSD17B10 Q99714 2/20 0.35
TSHR P16473 2/20 0.34
KMT2A Q03164 5/20 0.33
MEN1 O00255 3/20 0.33
HTT P42858 2/20 0.33
GAA P10253 1/20 0.33
TP53 P04637 1/20 0.32
LMNA P02545 2/20 0.32
TDP1 Q9NUW8 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
SIRT6 Q8N6T7 1/20 0.31
POLB P06746 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8062771 0.85 ALDH1A1 (0.36) ALDH1A1KDM4EMAPTHSD17B10TSHR
SCHEMBL8056365 0.78 ALDH1A1 (0.37) ALDH1A1KDM4EMAPTHSD17B10TSHR
SCHEMBL8062746 0.77 RXRA (0.36) ALDH1A1KDM4EMAPTHSD17B10TSHR
SCHEMBL8058178 0.77 CASP3 (0.44) ALDH1A1KDM4EMAPTHSD17B10TSHR
SCHEMBL8062776 0.76 ALDH1A1 (0.34) ALDH1A1KDM4EMAPTHSD17B10TSHR
SCHEMBL8060726 0.76 TSHR (0.34) ALDH1A1KDM4EMAPTHSD17B10TSHR
SCHEMBL8057016 0.75 ALDH1A1 (0.35) ALDH1A1KDM4EMAPTHSD17B10TSHR
SCHEMBL8062982 0.75 ALDH1A1 (0.34) ALDH1A1KDM4EMAPTHSD17B10TSHR
SCHEMBL8058104 0.75 RARA (0.37) ALDH1A1KDM4EMAPTHSD17B10TSHR
SCHEMBL8056504 0.74 IRAK4 (0.35) ALDH1A1KDM4EMAPTHSD17B10TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed