SCHEMBL8060706

SCHEMBL8060706

NC(N)=NC(=O)c1ccc2c(c1)S(=O)(=O)CCO2

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 4/20 0.42
HTR7 P34969 2/20 0.42
TSHR P16473 1/20 0.41
DRD2 P14416 1/20 0.40
ADRA1D P25100 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8056208 0.86 HTR2B (0.44) HTR2BHTR7DRD2ADRA1DHTR2A
SCHEMBL8060888 0.79
SCHEMBL8056251 0.77 HTR2B (0.44) HTR2BHTR7DRD2ADRA1DHTR2A
SCHEMBL8058186 0.76 HTR7 (0.49) HTR2BHTR7DRD2ADRA1DHTR2A
SCHEMBL8060804 0.76 CYP2C9 (0.46) TSHR
SCHEMBL8058190 0.75 SLC9A1 (0.43) HTR2BHTR7
SCHEMBL8056214 0.75 SLC9A1 (0.46) HTR2BHTR7
SCHEMBL8057034 0.75 HTR2B (0.41) HTR2BHTR7DRD2ADRA1DHTR2A
SCHEMBL8057351 0.74
SCHEMBL8060753 0.74 HTR7 (0.47) HTR2BHTR7DRD2ADRA1DHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed