SCHEMBL8060804

SCHEMBL8060804

COC(=O)c1ccc2c(c1)S(=O)(=O)CCO2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.46
ALDH1A1 P00352 6/20 0.44
TSHR P16473 2/20 0.44
LMNA P02545 1/20 0.44
MAPK1 P28482 1/20 0.44
KDM4E B2RXH2 6/20 0.44
SMN1; SMN2 Q16637 4/20 0.44
NPC1 O15118 5/20 0.43
RAB9A P51151 5/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
CASP3 P42574 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
CA12 O43570 2/20 0.42
CA9 Q16790 2/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42
XDH P47989 1/20 0.42
CA14 Q9ULX7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29070078 0.92 CYP2C9 (0.45) CYP2C9ALDH1A1TSHRLMNAMAPK1
SCHEMBL8056514 0.85 NPC1 (0.45) CYP2C9ALDH1A1TSHRLMNAMAPK1
SCHEMBL8056203 0.80 ALDH1A1 (0.44) CYP2C9ALDH1A1TSHRLMNAMAPK1
SCHEMBL17957599 0.79 KEAP1 (0.52) CYP2C9ALDH1A1TSHRLMNAMAPK1
SCHEMBL668237 0.78 KDM4E (0.62) ALDH1A1TSHRLMNAMAPK1KDM4E
SCHEMBL8060706 0.76 HTR2B (0.42) TSHR
SCHEMBL8056485 0.75 CA12 (0.53) ALDH1A1KDM4ESMN1; SMN2NPC1RAB9A
SCHEMBL8057027 0.75 RAB9A (0.43) CYP2C9ALDH1A1LMNAKDM4ESMN1; SMN2
SCHEMBL8056280 0.75 KDM4E (0.43) ALDH1A1TSHRKDM4ESMN1; SMN2NPC1
SCHEMBL29070074 0.75 ALDH1A1 (0.46) ALDH1A1TSHRLMNAMAPK1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed