SCHEMBL8065083

SCHEMBL8065083

O=C(O)c1cc([N+](=O)[O-])c([N+](=O)[O-])c(Cl)c1Cl

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C19 P33261 1/20 0.53
DTYMK P23919 1/20 0.44
CDK2 P24941 1/20 0.43
TSHR P16473 5/20 0.42
GPR35 Q9HC97 1/20 0.42
CASP6 P55212 1/20 0.41
PKM P14618 1/20 0.41
APEX1 P27695 1/20 0.40
VCAM1 P19320 1/20 0.39
SLC25A1 P53007 1/20 0.38
CYP3A4 P08684 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3291904 0.86 ALDH1A1 (0.60) ALDH1A1CYP1A2CYP2D6CYP2C19DTYMK
SCHEMBL1478701 0.86 ALDH1A1 (0.60) ALDH1A1CYP1A2CYP2D6CYP2C19DTYMK
SCHEMBL12603011 0.85 GPR35 (0.53) ALDH1A1CYP1A2CYP2D6CYP2C19DTYMK
SCHEMBL29891185 0.81 ALDH1A1 (0.52) ALDH1A1CYP1A2CYP2D6CYP2C19DTYMK
SCHEMBL27081346 0.81 ALDH1A1 (0.52) ALDH1A1CYP1A2CYP2D6CYP2C19DTYMK
SCHEMBL10954250 0.81 VCAM1 (0.55) ALDH1A1CYP1A2CYP2C19CDK2TSHR
SCHEMBL29886620 0.81 ALDH1A1 (0.44) ALDH1A1CYP1A2CYP2D6CYP2C19DTYMK
SCHEMBL11799475 0.79 CASP6 (0.48) ALDH1A1CYP1A2CYP2D6CYP2C19DTYMK
SCHEMBL8744067 0.79 ALDH1A1 (0.54) ALDH1A1CYP1A2CYP2D6CYP2C19TSHR
SCHEMBL8063523 0.79 ALDH1A1 (0.49) ALDH1A1CYP1A2CYP2D6CYP2C19DTYMK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1016405-A2 Arylating medicaments Radopath Pharmaceuticals International Limited (GB) 2000-07-05 EP claimed
EP-0700287-A1 ARYLATING MEDICAMENTS RADOPATH LIMITED (GB) 1996-03-13 EP claimed
WO-1994027584-A2 ARYLATING MEDICAMENTS RADOPATH LIMITED (GB) 1994-12-08 WO claimed