SCHEMBL8065580

SCHEMBL8065580

CCc1ccc(-c2ccc(C(F)(F)F)cc2F)cc1CC.CN[C@@H](CS)C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 5/20 0.45
AKR1C2 P52895 5/20 0.45
APP P05067 2/20 0.45
PPARD Q03181 3/20 0.42
ALOX5AP P20292 7/20 0.38
FEN1 P39748 7/20 0.38
PPARG P37231 1/20 0.38
PPARA Q07869 1/20 0.38
FFAR1 O14842 1/20 0.37
RORC P51449 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8064698 0.88 MEN1 (0.42) AKR1C3AKR1C2APP
SCHEMBL8079616 0.88 MEN1 (0.42) AKR1C3AKR1C2APP
SCHEMBL8074686 0.87 PSEN1 (0.42) AKR1C3AKR1C2PPARDPPARAFFAR1
SCHEMBL8064602 0.85 APP (0.40) AKR1C3AKR1C2APP
SCHEMBL8072952 0.85 APP (0.40) AKR1C3AKR1C2APP
SCHEMBL8078804 0.85 SLC1A3 (0.46) AKR1C3AKR1C2
SCHEMBL8075216 0.84 ACMSD (0.40) AKR1C3AKR1C2PPARGPPARAFFAR1
SCHEMBL8074144 0.84 ACMSD (0.40) AKR1C3AKR1C2PPARGPPARAFFAR1
SCHEMBL8080386 0.83 AKR1C3 (0.49) AKR1C3AKR1C2APP
SCHEMBL8080154 0.81 PPARG (0.41) AKR1C3AKR1C2PPARGPPARAFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999034790-A1 GLYCINE TRANSPORT INHIBITORS ALLELIX NEUROSCIENCE, INC. (US) 1999-07-15 WO claimed
US-6166072-A Amino acid derivatives ALLELIX NEUROSCIENCE, INC. (CA) 2000-12-26 US disclosed
WO-1999034790-A1 GLYCINE TRANSPORT INHIBITORS ALLELIX NEUROSCIENCE, INC. (US) 1999-07-15 WO disclosed