SCHEMBL8066360

SCHEMBL8066360

O=S(=O)(Nc1nc(-c2ccccc2)c(-c2ccccc2)s1)C(F)(F)F

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CDC25B P30305 10/20 0.59
DUSP3 P51452 10/20 0.59
PTPN1 P18031 9/20 0.59
KDM1A O60341 1/20 0.55
PTGS2 P35354 3/20 0.51
XIAP P98170 1/20 0.47
HSD17B10 Q99714 1/20 0.46
ALDH1A1 P00352 2/20 0.45
MAPT P10636 2/20 0.45
KMT2A Q03164 2/20 0.45
MEN1 O00255 1/20 0.45
RORC P51449 1/20 0.45
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C19 P33261 1/20 0.44
HPGD P15428 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
PTGS1 P23219 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8056899 0.94 PTPN1 (0.54) CDC25BDUSP3PTPN1KDM1APTGS2
SCHEMBL8066039 0.92 CDC25B (0.53) CDC25BDUSP3PTPN1KDM1APTGS2
SCHEMBL9615924 0.92 KDM1A (0.58) CDC25BDUSP3PTPN1KDM1APTGS2
SCHEMBL8067396 0.90 MAPT (0.61) CDC25BDUSP3PTPN1KDM1APTGS2
SCHEMBL8056502 0.90 MAPT (0.61) CDC25BDUSP3PTPN1KDM1APTGS2
SCHEMBL8060240 0.88 PTPN1 (0.64) CDC25BDUSP3PTPN1KDM1APTGS2
SCHEMBL8072543 0.87 PTGS2 (0.51) CDC25BDUSP3PTPN1KDM1APTGS2
SCHEMBL8067403 0.84 MAPT (0.60) CDC25BDUSP3PTPN1PTGS2ALDH1A1
SCHEMBL4115163 0.81 HSD17B10 (0.68) CDC25BDUSP3PTPN1KDM1APTGS2
SCHEMBL4110122 0.79 KDM1A (0.76) CDC25BDUSP3PTPN1KDM1APTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0592664-B1 DERIVATIVES OF DIPHENYLTHIAZOLE WITH ANTIINFLAMMATORY ACTIVITY HISAMITSU PHARMACEUTICAL CO (JP) 2000-07-05 EP claimed
US-5449783-A Antiinflammatory, analgesic, antiallergic, diuretic agents, anticoagulants HISAMITSU PHARMACEUTICAL CO., INC. (JP) 1995-09-12 US claimed
JP-3173876-A None JP disclosed
EP-0592664-B1 DERIVATIVES OF DIPHENYLTHIAZOLE WITH ANTIINFLAMMATORY ACTIVITY HISAMITSU PHARMACEUTICAL CO (JP) 2000-07-05 EP disclosed
US-5449783-A Antiinflammatory, analgesic, antiallergic, diuretic agents, anticoagulants HISAMITSU PHARMACEUTICAL CO., INC. (JP) 1995-09-12 US disclosed
EP-0592664-A1 NOVEL DIPHENYLTHYAZOLE DERIVATIVE Hisamitsu Pharmaceutical Co., Inc. (JP) 1994-04-20 EP disclosed
JP-H03173876-A NEW DIPHENYLTHIAZOLE DERIVATIVE HISAMITSU PHARMACEUT CO INC 1991-07-29 JP disclosed