SCHEMBL8066632

SCHEMBL8066632

O=[N+]([O-])c1cc(Cl)cc(Cl)c1[N+](=O)[O-]

nearest known ligand 0.75

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.75
TSHR P16473 3/20 0.75
MAPK1 P28482 2/20 0.55
VCAM1 P19320 5/20 0.43
GRIN2D O15399 1/20 0.42
GRIN3B O60391 1/20 0.42
GRIN1 Q05586 1/20 0.42
GRIN2A Q12879 1/20 0.42
GRIN2B Q13224 1/20 0.42
GRIN2C Q14957 1/20 0.42
GRIN3A Q8TCU5 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
GPR35 Q9HC97 2/20 0.41
CYP3A4 P08684 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
TTR P02766 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11800281 0.89 TSHR (0.62) ALDH1A1TSHRMAPK1VCAM1TDP1
SCHEMBL954217 0.86 ALDH1A1 (1.00) ALDH1A1TSHRMAPK1GRIN2DGRIN3B
SCHEMBL11793608 0.81 GPR35 (0.63) ALDH1A1TSHRMAPK1TDP1GPR35
SCHEMBL11804756 0.80 ALDH1A1 (0.58) ALDH1A1TSHRMAPK1VCAM1TDP1
SCHEMBL6186068 0.80 ALDH1A1 (0.58) ALDH1A1TSHRMAPK1VCAM1TDP1
SCHEMBL31694394 0.78 ALDH1A1 (0.56) ALDH1A1TSHRMAPK1VCAM1GRIN2D
SCHEMBL25422898 0.77 ALDH1A1 (0.54) ALDH1A1TSHRMAPK1VCAM1TDP1
SCHEMBL310420 0.77 GPR35 (0.69) ALDH1A1TSHRMAPK1TDP1GPR35
SCHEMBL204939 0.77 ALDH1A1 (0.55) ALDH1A1TSHRMAPK1VCAM1TDP1
SCHEMBL11138337 0.77 ALDH1A1 (0.72) ALDH1A1TSHRMAPK1GRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1016405-A2 Arylating medicaments Radopath Pharmaceuticals International Limited (GB) 2000-07-05 EP claimed
CN-1124012-A Arylating medicaments RADOPATH LTD (GB) 1996-06-05 CN claimed
EP-0700287-A1 ARYLATING MEDICAMENTS RADOPATH LIMITED (GB) 1996-03-13 EP claimed
WO-1994027584-A2 ARYLATING MEDICAMENTS RADOPATH LIMITED (GB) 1994-12-08 WO claimed
EP-1016405-A2 Arylating medicaments Radopath Pharmaceuticals International Limited (GB) 2000-07-05 EP disclosed
US-5574188-A NITRATING DICHLOROBENZENE, DIBENZYLOXY INTERMEDIATE, MULTISTEP BAYER AKTIENGESELLSCHAFT (DE) 1996-11-12 US disclosed
CN-1124012-A Arylating medicaments RADOPATH LTD (GB) 1996-06-05 CN disclosed
EP-0325892-B1 PROCESS FOR THE PREPARATION OF HALOGENATED PRIMARY AMINES CIBA-GEIGY AG (CH) 1993-02-03 EP disclosed
EP-0473552-A1 Process for the preparation of halogenated aromatic primary amines CIBA-GEIGY AG (CH) 1992-03-04 EP disclosed
US-4960936-A Process for the preparation of halogenated aromatic primary amines CIBA-GEIGY CORPORATION (US) 1990-10-02 US disclosed
EP-0325892-A2 Process for the preparation of halogenated primary amines CIBA-GEIGY AG (CH) 1989-08-02 EP disclosed
US-4102924-A REACTING ACYLAMINO-ARYLS WITH HALO-ARYLS BAYER AKTIENGESELLSCHAFT (DE) 1978-07-25 US disclosed
US-4080491-A CATALYST CONTAINS ORGANOMETALLIC COMPOUND AND THE REACTION PRODUCT OF TUNGSTEN OR MOLYBDENUM OXIDE AND A PHOSPHOROUS HALIDE OR OXYHALIDE SHOWA DENKO K.K. (JA) 1978-03-21 US disclosed