SCHEMBL8066700

SCHEMBL8066700

COc1cccc(C2CCCC/C2=C/c2nc(-c3ccccc3)c(-c3ccccc3)o2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GID4 Q8IVV7 1/20 0.43
KDM4E B2RXH2 3/20 0.41
HTT P42858 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
LMNA P02545 1/20 0.41
RECQL P46063 1/20 0.41
RXRA P19793 3/20 0.40
RXRB P28702 3/20 0.40
NR4A2 P43354 3/20 0.36
RXRG P48443 1/20 0.36
MAPT P10636 2/20 0.36
HPGD P15428 1/20 0.36
DDB1 Q16531 1/20 0.36
CRBN Q96SW2 1/20 0.36
PTGIR P43119 2/20 0.36
CASP3 P42574 1/20 0.36
RAB9A P51151 1/20 0.36
SENP8 Q96LD8 1/20 0.36
SENP7 Q9BQF6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8066704 1.00 GID4 (0.43) GID4KDM4EHTTTDP1SMN1; SMN2
SCHEMBL9006849 0.88 NR4A2 (0.42) KDM4EHTTTDP1SMN1; SMN2LMNA
SCHEMBL9006842 0.87 NR4A2 (0.41) KDM4EHTTTDP1SMN1; SMN2LMNA
SCHEMBL8065993 0.86 FABP4 (0.50) KDM4EHPGDPTGIRMEN1KMT2A
SCHEMBL8065990 0.86 FABP4 (0.50) KDM4EHPGDPTGIRMEN1KMT2A
SCHEMBL8055531 0.82 PTGIR (0.47) KDM4EHTTTDP1SMN1; SMN2LMNA
SCHEMBL8055530 0.82 PTGIR (0.47) KDM4EHTTTDP1SMN1; SMN2LMNA
SCHEMBL9006916 0.73 RXRA (0.41) KDM4ELMNARXRARXRBNR4A2
SCHEMBL8065136 0.73 KDM4E (0.44) GID4KDM4EHTTTDP1SMN1; SMN2
SCHEMBL8074838 0.72 KDM4E (0.46) KDM4EHTTTDP1SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0736018-B1 4,5-DIARYLOXAZOLE DERIVATIVES FUJISAWA PHARMACEUTICAL CO (JP) 2000-07-05 EP disclosed
US-6025375-A INHIBITORY ACTIVITY ON PLATELET AGGREGATION, VASODILATING ACTIVITY, ANTIHYPERTENSIVE ACTIVITY OR THE LIKE AND ARE PROSTAGLANDIN I.SUB.2 AGONISTS, FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-02-15 US disclosed
WO-1995017393-A1 4,5-DIARYLOXAZOLE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-06-29 WO disclosed