SCHEMBL8067464

SCHEMBL8067464

CCOC(=O)CNC=CC(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.44
MGAM O43451 1/20 0.39
SI P14410 1/20 0.39
MGAM2 Q2M2H8 1/20 0.39
CTSK P43235 1/20 0.38
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
HTT P42858 2/20 0.37
CYP1A2 P05177 1/20 0.37
SMN1; SMN2 Q16637 4/20 0.36
LMNA P02545 1/20 0.35
NR1I2 O75469 1/20 0.35
PGR P06401 1/20 0.35
CYP3A4 P08684 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
SLC6A2 P23975 1/20 0.35
TBXAS1 P24557 1/20 0.35
DRD3 P35462 1/20 0.35
OPRK1 P41145 1/20 0.35
PDE4D Q08499 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8746791 0.80 ALDH1A1 (0.37) GAACYP2C9CYP2C19CYP1A2SMN1; SMN2
SCHEMBL8488938 0.76 ADH1B (0.35) GAACTSKCYP2C9CYP2C19HTT
SCHEMBL1366125 0.75 HCAR2 (0.59) CYP2C9CYP2C19HTTLMNANR1I2
SCHEMBL1366123 0.75 HCAR2 (0.59) CYP2C9CYP2C19HTTLMNANR1I2
SCHEMBL8093037 0.75 GAA (0.39) GAAMGAMSIMGAM2CYP2C9
SCHEMBL12274267 0.73 CA2 (0.38) CTSKCYP2D6
SCHEMBL28682778 0.72 HTT (0.38) GAAMGAMSIMGAM2CTSK
SCHEMBL28383745 0.72 HTT (0.38) GAAMGAMSIMGAM2CTSK
SCHEMBL7437449 0.72 GAA (0.48) GAAMGAMSIMGAM2CTSK
SCHEMBL1936376 0.72 ALDH1A1 (0.52) GAAMGAMSIMGAM2CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6069272-A Simplified method for the production of vinyl glycine (2-aminobut-3-enoic acid) and a convenient resolution of a derivative HOECHST AKTIENGESELLSCHAFT (DE) 2000-05-30 US disclosed
EP-0559927-B1 A simplified method for the production of vinyl glycine (2-aminobut-3-enioc acid) and a convenient resolution of a derivative HOECHST AG (DE) 1997-03-05 EP disclosed
EP-0559927-A1 A simplified method for the production of vinyl glycine (2-aminobut-3-enioc acid) and a convenient resolution of a derivative Hoechst Schering AgrEvo GmbH (DE) 1993-09-15 EP disclosed