SCHEMBL8068014

SCHEMBL8068014

O=C(/C=C/c1ccncc1)C12CC3CC(CC(C3)C1)C2

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
JUN P05412 1/20 0.51
NFKB1 P19838 1/20 0.51
CYP17A1 P05093 7/20 0.48
CYP19A1 P11511 5/20 0.48
KMT2A Q03164 3/20 0.48
ALDH1A1 P00352 3/20 0.48
MEN1 O00255 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.44
HSD11B1 P28845 1/20 0.43
LMNA P02545 2/20 0.42
HTT P42858 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
POLB P06746 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
EPHX2 P34913 1/20 0.42
KDM4E B2RXH2 1/20 0.42
TDP1 Q9NUW8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6092331 1.00 JUN (0.51) JUNNFKB1CYP17A1CYP19A1KMT2A
SCHEMBL6091145 0.84 GABBR2 (0.53) KMT2AALDH1A1MEN1LMNAHTT
SCHEMBL12040547 0.84 GABBR2 (0.53) KMT2AALDH1A1MEN1LMNAHTT
SCHEMBL622342 0.84 CYP17A1 (0.50) CYP17A1CYP19A1KMT2AALDH1A1MEN1
SCHEMBL1769996 0.82 MAPT (0.56) JUNNFKB1CYP17A1CYP19A1KMT2A
SCHEMBL8077622 0.82 MAPT (0.56) JUNNFKB1CYP17A1CYP19A1KMT2A
SCHEMBL6092094 0.81 HSD11B1 (0.51) KMT2AALDH1A1MEN1HSD11B1LMNA
SCHEMBL18317450 0.81 ALDH1A1 (0.45) KMT2AALDH1A1MEN1LMNAHTT
SCHEMBL18325433 0.81 ALDH1A1 (0.45) KMT2AALDH1A1MEN1LMNAHTT
SCHEMBL6090902 0.81 CYP1A2 (0.51) KMT2AALDH1A1MEN1L3MBTL1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640072-B1 Derivatives of pyridine as hydroxylase and lyase inhibitors BTG INT LTD (GB) 2000-08-23 EP disclosed
US-5595995-A ANTICARCINOGENIC AGENTS BRITISH TECHNOLOGY GROUP LIMITED (GB) 1997-01-21 US disclosed
EP-0640072-A1 SUBSTITUTED PYRIDINES, THEIR PREPARATION AND PHARMACEUTICAL USE BTG INTERNATIONAL LIMITED (GB) 1995-03-01 EP disclosed
WO-1993023375-A1 SUBSTITUTED PYRIDINES, THEIR PREPARATION AND PHARMACEUTICAL USE BRITISH TECHNOLOGY GROUP LIMITED (GB) 1993-11-25 WO disclosed