SCHEMBL8068053

SCHEMBL8068053

C=C(C)C(=O)OCCOCCNc1ccc2c(c1)Cc1ccccc1-2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.51
ADRA2A P08913 1/20 0.51
MAOA P21397 1/20 0.51
SLC6A2 P23975 1/20 0.51
HTR2C P28335 1/20 0.51
SLC6A4 P31645 1/20 0.51
HTR2B P41595 1/20 0.51
RAB9A P51151 5/20 0.47
NPC1 O15118 4/20 0.47
KDM4E B2RXH2 4/20 0.44
LMNA P02545 3/20 0.44
TDP1 Q9NUW8 1/20 0.44
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
MAPT P10636 6/20 0.43
ALDH1A1 P00352 3/20 0.43
HPGD P15428 2/20 0.43
MAPK1 P28482 2/20 0.43
CYP3A4 P08684 1/20 0.41
SLC1A3 P43003 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21950454 0.82 CYP1A2 (0.56) CYP1A2ADRA2AMAOASLC6A2HTR2C
SCHEMBL8053871 0.79 ALDH1A1 (0.44) CYP1A2RAB9ANPC1KDM4ELMNA
SCHEMBL8068096 0.78 THRB (0.42) CYP1A2RAB9ANPC1KDM4ELMNA
SCHEMBL13144122 0.77 MAPT (0.51) CYP1A2MAOARAB9ANPC1TDP1
Fluorene SCHEMBL19019691 0.73 GABRP (0.52) CYP1A2ADRA2AMAOASLC6A2HTR2C
SCHEMBL4443581 0.72 CYP1A2 (0.74) CYP1A2ADRA2AMAOASLC6A2HTR2C
SCHEMBL8053806 0.72 THRB (0.43) CYP1A2RAB9ANPC1KDM4EMEN1
SCHEMBL305728 0.71 POLB (0.44) KDM4ETDP1MAPTALDH1A1TSHR
SCHEMBL27294859 0.71 MEN1 (0.51) MAOARAB9ANPC1LMNAMEN1
Fluorene SCHEMBL608981 0.71 ALDH1A1 (0.52) CYP1A2ADRA2AMAOASLC6A2HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5948268-A DISSOLVING IN WATER TO BE TREATED A POLYMER FORMED FROM WATER SOLUBLE MONOMER UNITS COMPRISING A (POLY)ALKYLENE OXIDE END CAPPED WITH AN ADDITION POLYMERIZABLE GROUP AT ONE END AND AN INTENSELY FLUORESCENT GROUP AT OTHER NIPPON SHOKUBAI CO., LTD. (JP) 1999-09-07 US claimed
EP-0761604-B1 An agent for water treatment NIPPON CATALYTIC CHEM IND (JP) 2000-06-14 EP disclosed
US-5948268-A DISSOLVING IN WATER TO BE TREATED A POLYMER FORMED FROM WATER SOLUBLE MONOMER UNITS COMPRISING A (POLY)ALKYLENE OXIDE END CAPPED WITH AN ADDITION POLYMERIZABLE GROUP AT ONE END AND AN INTENSELY FLUORESCENT GROUP AT OTHER NIPPON SHOKUBAI CO., LTD. (JP) 1999-09-07 US disclosed
EP-0761604-A2 An agent for water treatment NIPPON SHOKUBAI CO., LTD. (JP) 1997-03-12 EP disclosed