SCHEMBL8068944

SCHEMBL8068944

COc1ccc(CN2CC3C(C2)C3c2ccccc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.62
HRH2 P25021 1/20 0.53
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
DRD4 P21917 2/20 0.50
DRD2 P14416 1/20 0.50
DRD3 P35462 1/20 0.50
PAX8 Q06710 1/20 0.49
FAAH O00519 1/20 0.49
ALDH1A1 P00352 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12489466 0.92 PAX8 (0.56) SIGMAR1HRH2DRD4PAX8ALDH1A1
SCHEMBL12488080 0.92 PAX8 (0.56) SIGMAR1HRH2DRD4PAX8ALDH1A1
SCHEMBL12488076 0.92 PAX8 (0.56) SIGMAR1HRH2DRD4PAX8ALDH1A1
SCHEMBL12488083 0.92 PAX8 (0.56) SIGMAR1HRH2DRD4PAX8ALDH1A1
SCHEMBL19559108 0.82 SIGMAR1 (0.51) SIGMAR1HRH2MEN1KMT2ADRD4
SCHEMBL7072989 0.82 FUCA1 (0.55) SIGMAR1ALDH1A1
SCHEMBL4877680 0.82 FAAH (0.53) SIGMAR1KMT2APAX8FAAHALDH1A1
SCHEMBL13602414 0.80 SIGMAR1 (0.47) SIGMAR1HRH2MEN1KMT2ADRD2
SCHEMBL6572711 0.80 SIGMAR1 (0.64) SIGMAR1HRH2MEN1KMT2ADRD4
SCHEMBL14197151 0.80 LMNA (0.54) SIGMAR1KMT2AFAAHALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6096755-A N-substituted azabicycloalkane derivatives, their preparation and use BASF AKTIENGESELLSCHAFT (DE) 2000-08-01 US disclosed
EP-0731802-A1 N-SUBSTITUTED AZABICYCLOALKANE DERIVATIVES AS NEUROLEPTIKA ASF BASF AKTIENGESELLSCHAFT (DE) 1996-09-18 EP disclosed
WO-1996026978-A1 IMPROVED SELF-LUBRICATING THERMOPLASTIC POLYMER COMPOSITION HOECHST CELANESE CORPORATION (US) 1996-09-06 WO disclosed
EP-0728136-A1 N-SUBSTITUTED AZABICYCLOALKANE DERIVATIVES, THEIR PREPARATION AND USE BASF AKTIENGESELLSCHAFT (DE) 1996-08-28 EP disclosed
WO-1995015327-A1 N-SUBSTITUTED AZABICYCLOALKANE DERIVATIVES AS NEUROLEPTIKA ASF BASF AKTIENGESELLSCHAFT (DE) 1995-06-08 WO disclosed
WO-1995013279-A1 N-SUBSTITUTED AZABICYCLOALKANE DERIVATIVES, THEIR PREPARATION AND USE BASF AKTIENGESELLSCHAFT (DE) 1995-05-18 WO disclosed