SCHEMBL8069504

SCHEMBL8069504

COc1ccc2c(c1)nc(Cl)n2-c1cnc(NC(=O)c2c(C)cccc2F)cn1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
STIM1 Q13586 1/20 0.46
ORAI1 Q96D31 1/20 0.46
ORAI2 Q96SN7 1/20 0.46
LCK P06239 1/20 0.40
RAB9A P51151 2/20 0.39
GRM5 P41594 1/20 0.39
NPC1 O15118 1/20 0.39
CYP1A2 P05177 1/20 0.39
IL2 P60568 4/20 0.37
MEN1 O00255 1/20 0.37
POLB P06746 1/20 0.37
KMT2A Q03164 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
ABL1 P00519 1/20 0.37
RORC P51449 3/20 0.36
BRPF1 P55201 1/20 0.36
SCN9A Q15858 1/20 0.36
BRD4 O60885 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3104227 0.95 RAB9A (0.44) STIM1ORAI1ORAI2RAB9AGRM5
SCHEMBL8069094 0.91 STIM1 (0.43) STIM1ORAI1ORAI2LCKRAB9A
SCHEMBL3103400 0.87 RAB9A (0.45) RAB9AGRM5NPC1CYP1A2IL2
SCHEMBL647154 0.83 RAB9A (0.43) RAB9ANPC1CYP1A2IL2MEN1
SCHEMBL647823 0.77 RET (0.36) RAB9AGRM5NPC1CYP1A2MEN1
SCHEMBL8062134 0.77 STIM1 (0.44) STIM1ORAI1ORAI2IL2MEN1
SCHEMBL8070992 0.76 STIM1 (0.44) STIM1ORAI1ORAI2LCKIL2
SCHEMBL10151672 0.76 RAB9A (0.44) RAB9AGRM5NPC1CYP1A2IL2
SCHEMBL646105 0.76 RAB9A (0.43) RAB9ANPC1CYP1A2IL2MEN1
SCHEMBL648258 0.76 STIM1 (0.36) STIM1ORAI1RAB9AGRM5NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009038775-A1 SUBSTITUTED BENZOIMIDAZOLYL-PYRAZINE COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES SYNTA PHARMACEUTICALS CORP. (US) 2009-03-26 WO disclosed