SCHEMBL807059

SCHEMBL807059

COc1ncc(-c2ccc3nc(N)c(C(=O)N4CCCCC4)cc3c2)cc1N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3C3 Q8NEB9 1/20 0.46
HPGD P15428 9/20 0.44
TDP1 Q9NUW8 1/20 0.41
MAPT P10636 1/20 0.41
CASP1 P29466 1/20 0.41
GAK O14976 1/20 0.41
AURKA O14965 1/20 0.40
TTK P33981 1/20 0.40
AURKB Q96GD4 1/20 0.40
INCENP Q9NQS7 1/20 0.40
RAB9A P51151 2/20 0.40
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10274836 0.91 KCNH2 (0.48) PIK3C3HPGDMAPTCASP1AURKA
SCHEMBL807061 0.90 ATR (0.43) PIK3C3MAPTCASP1AURKATTK
SCHEMBL806763 0.90 KIT (0.49) PIK3C3HPGDMAPTGAKRAB9A
SCHEMBL807240 0.80 PIK3CG (0.67) PI4KAPIK3CG
SCHEMBL10274839 0.77 MAPT (0.56) MAPTCASP1AURKATTKAURKB
SCHEMBL789820 0.77 ALDH1A1 (0.43) PIK3C3HPGDTDP1RAB9AKDM4E
SCHEMBL807455 0.74 PI4KA (0.55) PI4KAPIK3CG
SCHEMBL807470 0.73 PIK3CG (0.55) PI4KAPIK3CG
SCHEMBL806791 0.73 PI4KA (0.43) PIK3C3HPGDRAB9AKDM4EALDH1A1
SCHEMBL789777 0.73 PIK3CG (0.66) PI4KAPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed