SCHEMBL8071055

SCHEMBL8071055

COC(=O)c1cc(N)c(-c2ccccc2)cc1C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.51
HSD17B10 Q99714 2/20 0.51
CFTR P13569 1/20 0.51
HPGD P15428 4/20 0.51
MAPT P10636 4/20 0.51
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
GAA P10253 2/20 0.51
GABRA1 P14867 2/20 0.48
GABRG2 P18507 2/20 0.48
GABRB3 P28472 2/20 0.48
GABRA3 P34903 2/20 0.48
LMNA P02545 1/20 0.48
PRKCZ Q05513 1/20 0.48
EGFR P00533 1/20 0.48
KDM4E B2RXH2 3/20 0.47
GLA P06280 1/20 0.47
CASP1 P29466 1/20 0.47
CASP7 P55210 1/20 0.47
ATM Q13315 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8068448 0.83 GABRA1 (0.49) ALDH1A1HPGDMAPTMEN1KMT2A
SCHEMBL12117486 0.82 ALDH1A1 (0.51) ALDH1A1HSD17B10CFTRHPGDMAPT
SCHEMBL27717289 0.82 ALDH1A1 (0.51) ALDH1A1HSD17B10CFTRHPGDMAPT
SCHEMBL16419694 0.80 GABRA1 (0.55) ALDH1A1HPGDMAPTMEN1KMT2A
SCHEMBL8059705 0.78 CFTR (0.53) ALDH1A1CFTRHPGDMAPTMEN1
SCHEMBL8608047 0.78 PTGS2 (0.52) ALDH1A1HPGDMAPTMEN1KMT2A
SCHEMBL1720999 0.78 KDM4E (0.56) ALDH1A1HSD17B10CFTRHPGDMAPT
SCHEMBL23628969 0.78 PTGS2 (0.58) ALDH1A1HSD17B10CFTRHPGDMAPT
SCHEMBL2686505 0.78 EGFR (0.61) ALDH1A1HSD17B10HPGDMAPTMEN1
SCHEMBL5799055 0.77 PTGS2 (0.48) ALDH1A1HSD17B10CFTRHPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057322-A USEFUL IN TREATMENT OF CARDIOVASCULAR DISEASES HOECHST AKTIENGESELLSCHAFT (DE) 2000-05-02 US disclosed