SCHEMBL8071504

SCHEMBL8071504

COc1ccc(CN2CCOCC2)nc1-c1cccc(NO)c1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 1/20 0.46
PDE4B Q07343 4/20 0.44
ALDH1A1 P00352 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
HSD17B10 Q99714 1/20 0.43
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.42
ADORA2A P29274 1/20 0.42
SLC2A1 P11166 1/20 0.41
HTT P42858 1/20 0.41
NPC1 O15118 1/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
RAB9A P51151 1/20 0.40
JAK2 O60674 1/20 0.40
JAK1 P23458 1/20 0.40
TYK2 P29597 1/20 0.40
JAK3 P52333 1/20 0.40
ALOX15 P16050 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8070648 0.80 PDE4B (0.42) PDE4BALDH1A1SMN1; SMN2NPC1LMNA
SCHEMBL3794467 0.80 PDE4B (0.60) CXCR4PDE4BSMN1; SMN2MAPTNPC1
SCHEMBL8066164 0.79 PDE4B (0.44) PDE4BMAPT
SCHEMBL8024647 0.79 PDE4B (0.46) PDE4B
SCHEMBL8053232 0.75 PDE4B (0.45) PDE4B
SCHEMBL8028328 0.73 PDE4B (0.41) PDE4BMAPTTP53
SCHEMBL8071898 0.73 PDE4B (0.56) PDE4B
SCHEMBL8072345 0.73 PDE4B (0.46) PDE4BALDH1A1MAPT
SCHEMBL29604383 0.66 CXCR4 (1.00) CXCR4ALDH1A1SMN1; SMN2HSD17B10KDM4E
SCHEMBL22167005 0.66 CXCR4 (0.61) CXCR4ALDH1A1SMN1; SMN2NPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009067600-A2 BIARYL PDE4 INHIBITORS FOR TREATING INFLAMMATION DECODE GENETICS EHF (IS) 2009-05-28 WO disclosed