SCHEMBL8072083

SCHEMBL8072083

CCCc1nc(Cl)c(C=O)n1Cc1ccc(-c2ccccc2)c(-c2nnn[nH]2)c1

nearest known ligand 0.56

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GP6 Q9HCN6 1/20 0.56
AGTR2 P50052 8/20 0.53
AGTR1 P30556 8/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8172767 0.95 GP6 (0.63) GP6AGTR2AGTR1
SCHEMBL976 0.91 GP6 (0.64) GP6AGTR2AGTR1
SCHEMBL7175115 0.86 AGTR2 (0.49) GP6AGTR2AGTR1
SCHEMBL6536653 0.86 AGTR1 (0.57) AGTR2AGTR1
SCHEMBL860 0.86 GP6 (0.72) GP6AGTR2AGTR1
SCHEMBL7362569 0.84 AGTR2 (0.72) GP6AGTR2AGTR1
SCHEMBL8469323 0.82 AGTR1 (0.46) AGTR2AGTR1
SCHEMBL9198036 0.81 AGTR2 (0.58) GP6AGTR2AGTR1
SCHEMBL9030299 0.81 AGTR2 (0.56) GP6AGTR2AGTR1
SCHEMBL3427175 0.81 AGTR1 (0.64) AGTR2AGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1019048-A1 USE OF AN ANGIOTENSIN II RECEPTOR ANTAGONIST FOR THE PREPARATION OF DRUGS TO INCREASE THE SURVIVAL RATE OF RENAL TRANSPLANT PATIENTS Merck Sharp Dohme (Italia) S.P.A. (IT) 2000-07-19 EP claimed
WO-1999016437-A1 USE OF AN ANGIOTENSIN II RECEPTOR ANTAGONIST FOR THE PREPARATION OF DRUGS TO INCREASE THE SURVIVAL RATE OF RENAL TRANSPLANT PATIENTS MERCK SHARP DOHME (ITALIA) S.P.A. (IT) 1999-04-08 WO claimed