SCHEMBL8074041

SCHEMBL8074041

Cc1ccc(NC(=O)NC(c2ccccc2)C(NC(=O)Nc2ccc(C(F)(F)F)cc2)c2ccccc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FPR2 P25090 4/20 0.55
RAB9A P51151 3/20 0.54
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
MAPT P10636 2/20 0.54
HTT P42858 1/20 0.54
EPHX2 P34913 2/20 0.54
NPC1 O15118 2/20 0.51
CASR P41180 1/20 0.50
CCR3 P51677 1/20 0.48
HSD17B10 Q99714 1/20 0.48
IDH1 O75874 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
STING1 Q86WV6 1/20 0.46
KEAP1 Q14145 1/20 0.46
NFE2L2 Q16236 1/20 0.46
BAZ1A Q9NRL2 1/20 0.46
MTOR P42345 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8074038 1.00 FPR2 (0.55) FPR2RAB9AMEN1KMT2AMAPT
SCHEMBL8074018 0.92 FPR2 (0.57) FPR2RAB9AMEN1KMT2AMAPT
SCHEMBL8072202 0.92 FPR2 (0.57) FPR2RAB9AMEN1KMT2AMAPT
SCHEMBL8074023 0.92 FPR2 (0.57) FPR2RAB9AMEN1KMT2AMAPT
SCHEMBL8067540 0.89 LMNA (0.58) FPR2RAB9AMEN1KMT2AMAPT
SCHEMBL8070011 0.89 LMNA (0.58) FPR2RAB9AMEN1KMT2AMAPT
SCHEMBL8067545 0.89 LMNA (0.58) FPR2RAB9AMEN1KMT2AMAPT
SCHEMBL8067629 0.88 FPR2 (0.56) FPR2RAB9AMEN1KMT2AMAPT
SCHEMBL8067627 0.88 FPR2 (0.56) FPR2RAB9AMEN1KMT2AMAPT
SCHEMBL8073834 0.87 RAB9A (0.62) FPR2RAB9AMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6103761-A Agents acting at cholecystokinin receptors WARNER-LAMBERT COMPANY (US) 2000-08-15 US disclosed
US-5389682-A Appetite suppressants, anxiolytic agents, gastric acid inhibition WARNER-LAMBERT COMPANY (US) 1995-02-14 US disclosed
WO-1994006757-A1 AGENTS ACTING AT CHOLECYSTOKININ RECEPTORS WARNER-LAMBERT COMPANY (US) 1994-03-31 WO disclosed