SCHEMBL8075018

SCHEMBL8075018

CN(C)CCc1ccc(Oc2ccc(C(=O)NC(N)=NCl)cc2C(F)(F)F)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 3/20 0.43
SLC6A4 P31645 3/20 0.43
LPAR1 Q92633 1/20 0.42
LPAR5 Q9H1C0 1/20 0.42
SIRT1 Q96EB6 1/20 0.42
DRD2 P14416 1/20 0.38
DRD3 P35462 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
THRA P10827 1/20 0.38
THRB P10828 1/20 0.38
ROCK2 O75116 1/20 0.38
BRAF P15056 4/20 0.37
HDAC1 Q13547 3/20 0.36
HDAC3 O15379 2/20 0.36
HDAC4 P56524 2/20 0.36
HDAC7 Q8WUI4 2/20 0.36
HDAC2 Q92769 2/20 0.36
HDAC10 Q969S8 2/20 0.36
HDAC11 Q96DB2 2/20 0.36
HDAC8 Q9BY41 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8074970 0.90 SLC6A2 (0.45) SLC6A2SLC6A4LPAR1LPAR5SIRT1
Hydrochloric Acid SCHEMBL8070331 0.89 SLC6A2 (0.44) SLC6A2SLC6A4LPAR1LPAR5SIRT1
SCHEMBL8059455 0.86 HRH3 (0.40) SLC6A2SLC6A4DRD2DRD3HRH3
SCHEMBL8068477 0.83 DRD2 (0.38) SLC6A2SLC6A4DRD2DRD3HRH3
SCHEMBL8068627 0.81 LPAR1 (0.48) SLC6A2SLC6A4LPAR1LPAR5SIRT1
Hydrochloric Acid SCHEMBL8059587 0.78 SIRT1 (0.42) SLC6A2SLC6A4LPAR1LPAR5SIRT1
SCHEMBL8444238 0.78 SLC6A2 (0.41) SLC6A2SLC6A4LPAR1LPAR5SIRT1
SCHEMBL8428715 0.78 SIRT1 (0.46) SIRT1THRBROCK2KDM4EMAPT
Hydrochloric Acid SCHEMBL8070897 0.77 SLC6A2 (0.40) SLC6A2SLC6A4LPAR1LPAR5SIRT1
Hydrochloric Acid SCHEMBL8426168 0.77 SIRT1 (0.46) SIRT1THRBROCK2KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057322-A USEFUL IN TREATMENT OF CARDIOVASCULAR DISEASES HOECHST AKTIENGESELLSCHAFT (DE) 2000-05-02 US disclosed