SCHEMBL8075909

SCHEMBL8075909

O=C[C@@H](Cc1ccccc1)N1C(=O)c2ccccc2C1=O

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.61
GAA P10253 1/20 0.61
TDP1 Q9NUW8 1/20 0.60
POLB P06746 2/20 0.58
L3MBTL1 Q9Y468 2/20 0.58
SMN1; SMN2 Q16637 2/20 0.54
PKM P14618 1/20 0.54
AADAT Q8N5Z0 1/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
LMNA P02545 1/20 0.47
MAPT P10636 1/20 0.47
TSHR P16473 1/20 0.47
HSD11B1 P28845 1/20 0.46
HTT P42858 1/20 0.45
RECQL P46063 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
CASP3 P42574 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7829080 1.00 ALDH1A1 (0.61) ALDH1A1GAATDP1POLBL3MBTL1
SCHEMBL7284629 1.00 ALDH1A1 (0.61) ALDH1A1GAATDP1POLBL3MBTL1
SCHEMBL8283041 0.89 TDP1 (0.51) ALDH1A1GAATDP1POLBL3MBTL1
SCHEMBL8283049 0.87 CASP3 (0.50) ALDH1A1GAATDP1POLBL3MBTL1
SCHEMBL13937943 0.85 TDP1 (0.58) ALDH1A1GAATDP1POLBL3MBTL1
SCHEMBL7796562 0.85 TDP1 (0.58) ALDH1A1GAATDP1POLBL3MBTL1
SCHEMBL7797911 0.85 TDP1 (0.58) ALDH1A1GAATDP1POLBL3MBTL1
SCHEMBL12834925 0.83 ALDH1A1 (0.65) ALDH1A1GAATDP1POLBL3MBTL1
SCHEMBL28798215 0.80 TDP1 (0.47) ALDH1A1GAATDP1POLBL3MBTL1
SCHEMBL10588010 0.79 ALDH1A1 (0.61) ALDH1A1GAATDP1POLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE36718-E 3-AMINO-1-NITRO-4-PHENYL-2-BUTANOL DERIVATIVES KANEKA CORPORATION (JP) 2000-05-30 US disclosed
EP-0657415-B1 METHOD OF PRODUCING 3-AMINO-2-HYDROXY-4-PHENYL-BUTYRIC ACID DERIVATIVES AND 3-AMINO-1-NITRO-4-PHENYL-2-BUTANOL INTERMEDIATES KANEKA CORP (JP) 1999-09-08 EP disclosed
US-5616726-A AN 3-AMINO-1-NITRO-4-PHENYL-2-BUTANOL BY ADDING NITROMETHANE STEREOSELECTIVELY IN THE PRESENCE OF A BASE TO AN OPTICAL ACTIVE AMINOALDEHYDE; CHEMICAL INTERMEDIATES FOR DRUGS; E.G. THE ANTICARCINOGENIC AGENT, BESTATIN KANEKA CORPORATION (JP) 1997-04-01 US disclosed
EP-0657415-A1 OPTICALLY ACTIVE AMINO ALCOHOL DERIVATIVE AND PROCESS FOR PRODUCING THE SAME KANEKA CORPORATION (JP) 1995-06-14 EP disclosed