SCHEMBL8076818

SCHEMBL8076818

C=CCn1c(N)nc2c(ncn2Cc2ccccc2)c1=O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNP P00491 3/20 0.55
ALDH1A1 P00352 2/20 0.52
KDM4E B2RXH2 1/20 0.52
HPGD P15428 1/20 0.52
HSD17B10 Q99714 1/20 0.52
PDE4A P27815 2/20 0.48
PDE4B Q07343 2/20 0.48
PDE4C Q08493 2/20 0.48
PDE4D Q08499 2/20 0.48
ADORA2A P29274 5/20 0.48
PI4KA P42356 1/20 0.48
PI4K2B Q8TCG2 1/20 0.48
PI4K2A Q9BTU6 1/20 0.48
PI4KB Q9UBF8 1/20 0.48
CYP3A4 P08684 2/20 0.47
CYP2C19 P33261 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
HIF1A Q16665 1/20 0.47
PHLPP2 Q6ZVD8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8165314 0.77 PNP (0.56) PNPALDH1A1PDE4APDE4BPDE4C
SCHEMBL6359920 0.75 CDK1 (0.49) PNPALDH1A1KDM4EPDE4APDE4B
SCHEMBL6522309 0.74 PNP (0.52) PNPALDH1A1PDE4APDE4BPDE4C
SCHEMBL2780215 0.73 PNP (0.43) PNPALDH1A1KDM4EHPGDHSD17B10
SCHEMBL6272417 0.71 ALDH1A1 (0.66) PNPALDH1A1PDE4APDE4BPDE4C
SCHEMBL8610343 0.71 ALDH1A1 (0.47) ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL18249 0.71 PNP (1.00) PNP
SCHEMBL1980959 0.70 PNP (0.97) PNP
SCHEMBL1640041 0.70 PDE4A (0.69) PNPALDH1A1PDE4APDE4BPDE4C
SCHEMBL8076823 0.70 ADORA3 (0.42) PNPALDH1A1KDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1017394-A1 CYCLIN DEPENDENT KINASE INHIBITING PURINE DERIVATIVES CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 2000-07-12 EP disclosed
WO-1999002162-A9 CYCLIN DEPENDENT KINASE INHIBITING PURINE DERIVATIVES CANCER RES CAMPAIGN TECH (GB) 1999-07-29 WO disclosed
WO-1999002162-A1 CYCLIN DEPENDENT KINASE INHIBITING PURINE DERIVATIVES CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 1999-01-21 WO disclosed