SCHEMBL8076823

SCHEMBL8076823

C=CCn1c(N)nc2c(c1=O)NCN2Cc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 3/20 0.42
ADORA2A P29274 1/20 0.42
ADORA1 P30542 1/20 0.42
PKM P14618 1/20 0.42
HSD17B10 Q99714 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
TTR P02766 1/20 0.41
PDE5A O76074 1/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
PNP P00491 3/20 0.38
GAA P10253 1/20 0.37
DHFR P00374 1/20 0.37
LMNA P02545 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8165320 0.77 BRD4 (0.38) CYP2C19ALDH1A1PNPLMNAMEN1
SCHEMBL6359923 0.76 PNP (0.43) ADORA3PKMCYP3A4PDE5APDE4A
SCHEMBL2780222 0.74 MEN1 (0.37) PKMHSD17B10PDE5APDE4APDE4B
SCHEMBL4144591 0.73 HPRT1 (0.50) PNP
SCHEMBL8076818 0.70 PNP (0.55) ADORA3ADORA2AADORA1HSD17B10CYP3A4
SCHEMBL28852897 0.67 HSP90AA1 (0.40) HSD17B10ALDH1A1KDM4ELMNASMN1; SMN2
SCHEMBL2946378 0.65 CYP3A4 (0.61) ADORA3ADORA2AADORA1PKMCYP3A4
SCHEMBL4584939 0.65 CYP3A4 (0.61) ADORA3ADORA2AADORA1PKMCYP3A4
SCHEMBL9278710 0.65 HPRT1 (0.54) PNPMEN1KMT2A
SCHEMBL20343752 0.64 ADORA2A (0.39) ADORA3ADORA2AADORA1LMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1017394-A1 CYCLIN DEPENDENT KINASE INHIBITING PURINE DERIVATIVES CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 2000-07-12 EP disclosed
WO-1999002162-A9 CYCLIN DEPENDENT KINASE INHIBITING PURINE DERIVATIVES CANCER RES CAMPAIGN TECH (GB) 1999-07-29 WO disclosed
WO-1999002162-A1 CYCLIN DEPENDENT KINASE INHIBITING PURINE DERIVATIVES CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 1999-01-21 WO disclosed