SCHEMBL8077028

SCHEMBL8077028

CC1=C(n2ccc(O)cc2=O)c2cc([N+](=O)[O-])ccc2OC1(C)C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 2/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA7 P43166 1/20 0.35
MALT1 Q9UDY8 1/20 0.35
ALDH1A1 P00352 5/20 0.34
TDP1 Q9NUW8 2/20 0.34
CYP3A4 P08684 1/20 0.34
MAPT P10636 3/20 0.33
CASP3 P42574 2/20 0.33
PTPRC P08575 1/20 0.33
S100A4 P26447 1/20 0.33
CASP1 P29466 1/20 0.33
CASP4 P49662 1/20 0.33
CASP7 P55210 1/20 0.33
CASP9 P55211 1/20 0.33
CASP6 P55212 1/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33
MEN1 O00255 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8085063 0.85 CA9 (0.35) CA9CA1CA2CA7MALT1
SCHEMBL8085346 0.84 ALDH1A1 (0.38) CA9CA1CA2CA7MALT1
SCHEMBL8085417 0.82 MALT1 (0.37) CA9CA1CA2CA7MALT1
SCHEMBL8084426 0.82 ALDH1A1 (0.36) CA9CA1CA2CA7MALT1
SCHEMBL8085086 0.81 MALT1 (0.35) MALT1MAPTCASP3LMNA
SCHEMBL8085151 0.81 MAPT (0.34) ALDH1A1MAPT
SCHEMBL8077225 0.81 HSD17B1 (0.35) ALDH1A1MAPTS100A4KMT2APOLB
SCHEMBL8084362 0.80 KDM4E (0.34) ALDH1A1MAPTTSHRKMT2APOLB
SCHEMBL8085089 0.80 MEN1 (0.37) CA9CA1CA2CA7MALT1
SCHEMBL8088427 0.80 MAPT (0.33) ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
US-5013853-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-05-07 US disclosed
EP-0340718-A1 Chroman derivatives MERCK PATENT GmbH (DE) 1989-11-08 EP disclosed