SCHEMBL8085346

SCHEMBL8085346

CC1=C(n2ccccc2=O)c2cc([N+](=O)[O-])ccc2OC1(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
PTPRC P08575 3/20 0.37
S100A4 P26447 2/20 0.37
BCHE P06276 1/20 0.37
ACHE P22303 1/20 0.37
CES1 P23141 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
MALT1 Q9UDY8 1/20 0.36
MAPT P10636 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36
POLB P06746 1/20 0.36
CYP3A4 P08684 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
CHRM2 P08172 1/20 0.35
HTR1A P08908 1/20 0.35
ADRA2A P08913 1/20 0.35
DRD1 P21728 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8184423 0.86 MALT1 (0.38) ALDH1A1PTPRCS100A4BCHEACHE
SCHEMBL8085417 0.86 MALT1 (0.37) ALDH1A1PTPRCS100A4BCHEACHE
SCHEMBL9734444 0.86 ALDH1A1 (0.36) ALDH1A1PTPRCS100A4BCHEACHE
SCHEMBL8090463 0.85 MALT1 (0.37) ALDH1A1PTPRCS100A4BCHEACHE
SCHEMBL9146508 0.85 CHRM2 (0.37) ALDH1A1PTPRCS100A4BCHEACHE
SCHEMBL9148573 0.85 ALDH1A1 (0.35) ALDH1A1PTPRCS100A4BCHEACHE
SCHEMBL9732962 0.85 MAPT (0.35) ALDH1A1PTPRCS100A4BCHEACHE
SCHEMBL10521128 0.84 KDM4E (0.36) ALDH1A1
SCHEMBL8077028 0.84 CA9 (0.35) ALDH1A1PTPRCS100A4MEN1KMT2A
SCHEMBL8077334 0.84 ALDH1A1 (0.38) ALDH1A1PTPRCS100A4BCHEACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5447943-A Smooth muscle relaxants or bronchodilators SYNTEX (U.S.A.) INC. (US) 1995-09-05 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
US-5250547-A Potassium channel activators; 5-lipoxygenase inhibitors; muscle relaxants; bronchodilators SYNTEX (U.S.A.) INC. (US) 1993-10-05 US disclosed
EP-0529654-A1 Benzopyran derivatives as potassium channel activators and 5-lipoxygenase inhibitors SYNTEX (U.S.A.) INC. (US) 1993-03-03 EP disclosed
US-5013853-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-05-07 US disclosed
EP-0340718-A1 Chroman derivatives MERCK PATENT GmbH (DE) 1989-11-08 EP disclosed