SCHEMBL8077041

SCHEMBL8077041

CC1(C)C=C(n2cc(C(=O)O)ccc2=O)c2cc([N+](=O)[O-])ccc2O1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 2/20 0.42
CA12 O43570 1/20 0.42
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
GFER P55789 1/20 0.40
ESPL1 Q14674 1/20 0.39
TDP1 Q9NUW8 2/20 0.38
SRD5A2 P31213 1/20 0.36
RARA P10276 2/20 0.36
RARB P10826 2/20 0.36
RARG P13631 2/20 0.36
TP53 P04637 1/20 0.35
AKR1B1 P15121 1/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
TTR P02766 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8085035 0.88 ALDH1A1 (0.38) CA9MEN1KMT2ATDP1AKR1B1
SCHEMBL10698039 0.86 CA9 (0.36) CA9CA12MEN1KMT2ATDP1
SCHEMBL8077069 0.84 ALDH1A1 (0.35) CA9MEN1KMT2ATDP1CA1
SCHEMBL8077241 0.84 ALDH1A1 (0.36) CA9MEN1KMT2ATDP1CA1
SCHEMBL8090742 0.84 SMN1; SMN2 (0.41) MEN1KMT2ATDP1SMN1; SMN2
SCHEMBL8077161 0.81 PDE4A (0.40) RARARARBRARG
SCHEMBL8090686 0.80 CA9 (0.42) CA9CA12MEN1KMT2AGFER
SCHEMBL7268307 0.79 ALDH1A1 (0.39) CA9MEN1KMT2ATDP1CA1
SCHEMBL8088352 0.78 KDM4E (0.37) CA9CA12MEN1KMT2AGFER
SCHEMBL10695563 0.78 CA9 (0.36) CA9CA12MEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
EP-0273262-A2 Chroman derivatives MERCK PATENT GmbH (DE) 1988-07-06 EP disclosed