SCHEMBL8090686

SCHEMBL8090686

CC1=C(n2cc(C(=O)O)ccc2=O)c2cc([N+](=O)[O-])ccc2OC1(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 2/20 0.42
CA12 O43570 1/20 0.42
ESPL1 Q14674 1/20 0.40
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
GFER P55789 1/20 0.39
TDP1 Q9NUW8 1/20 0.37
SRD5A2 P31213 1/20 0.35
TP53 P04637 1/20 0.34
ALDH1A1 P00352 2/20 0.34
POLB P06746 1/20 0.34
PKM P14618 1/20 0.34
NPY1R P25929 1/20 0.34
NPY2R P49146 1/20 0.34
AKR1B1 P15121 1/20 0.34
PTPN7 P35236 1/20 0.34
PTPN22 Q9Y2R2 1/20 0.34
TSHR P16473 2/20 0.33
MALT1 Q9UDY8 1/20 0.33
CA1 P00915 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8085417 0.88 MALT1 (0.37) CA9MEN1KMT2ATDP1ALDH1A1
SCHEMBL8085063 0.86 CA9 (0.35) CA9CA12MEN1KMT2ATDP1
SCHEMBL8085054 0.84 ALDH1A1 (0.35) CA9MEN1KMT2ATDP1ALDH1A1
SCHEMBL8085089 0.84 MEN1 (0.37) CA9MEN1KMT2ATDP1ALDH1A1
SCHEMBL8077323 0.84 SMN1; SMN2 (0.40) MEN1KMT2ATDP1ALDH1A1POLB
SCHEMBL8090111 0.82 RARA (0.36) ALDH1A1MALT1
SCHEMBL8077041 0.80 CA9 (0.42) CA9CA12ESPL1MEN1KMT2A
SCHEMBL8085346 0.80 ALDH1A1 (0.38) CA9MEN1KMT2ATDP1ALDH1A1
SCHEMBL8090492 0.79 KDM4E (0.36) CA9CA12MEN1KMT2AGFER
SCHEMBL8077028 0.78 CA9 (0.35) CA9CA12MEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
US-5013853-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-05-07 US disclosed
EP-0340718-A1 Chroman derivatives MERCK PATENT GmbH (DE) 1989-11-08 EP disclosed