SCHEMBL807540

SCHEMBL807540

C[C@@H]1CN(Cc2cc(Nc3nc4cccnc4s3)nc(N[C@H]3CCNC3)c2)C[C@H](C)O1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITK Q08881 2/20 0.46
LCK P06239 1/20 0.42
AURKB Q96GD4 1/20 0.42
SSTR5 P35346 1/20 0.41
RORC P51449 1/20 0.38
DHODH Q02127 1/20 0.38
PRKCI P41743 7/20 0.37
ALK Q9UM73 1/20 0.35
POLB P06746 1/20 0.35
IRAK4 Q9NWZ3 1/20 0.34
MAOB P27338 2/20 0.34
HTR6 P50406 2/20 0.34
NPC1 O15118 2/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2395616 0.87 ITK (0.56) ITKLCKAURKBSSTR5RORC
SCHEMBL10286645 0.82 ITK (0.44) ITKLCKAURKBSSTR5RORC
SCHEMBL807946 0.81 ITK (0.58) ITKLCKAURKBSSTR5RORC
SCHEMBL807743 0.80 ITK (0.57) ITKLCKAURKBSSTR5RORC
SCHEMBL808093 0.80 ITK (0.61) ITKLCKAURKBSSTR5RORC
SCHEMBL807803 0.80 ITK (0.58) ITKLCKAURKBSSTR5RORC
SCHEMBL808096 0.79 ITK (0.51) ITKLCKAURKBSSTR5RORC
SCHEMBL10285825 0.78 ITK (0.58) ITKLCKAURKBSSTR5RORC
SCHEMBL808081 0.77 ITK (0.54) ITKLCKAURKBSSTR5RORC
SCHEMBL10285603 0.75 ITK (0.45) ITKLCKAURKBSSTR5RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035055-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-22 WO disclosed