SCHEMBL807803

SCHEMBL807803

C[C@@H]1CN(Cc2cc(Nc3nc4cccnc4s3)nc(N[C@H]3CCN(C(=O)OC(C)(C)C)C3)c2)C[C@H](C)O1

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITK Q08881 2/20 0.58
RORC P51449 1/20 0.41
DHODH Q02127 1/20 0.41
SSTR5 P35346 1/20 0.41
TBK1 Q9UHD2 8/20 0.40
LCK P06239 1/20 0.39
AURKB Q96GD4 1/20 0.39
USP30 Q70CQ3 3/20 0.39
ADORA3 P0DMS8 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA2B P29275 1/20 0.38
HCK P08631 2/20 0.38
BTK Q06187 2/20 0.38
BRD4 O60885 1/20 0.37
CCNA2 P20248 1/20 0.37
CDK2 P24941 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL807926 0.91 ITK (0.59) ITKRORCDHODHSSTR5TBK1
SCHEMBL807946 0.88 ITK (0.58) ITKRORCDHODHSSTR5LCK
SCHEMBL808093 0.87 ITK (0.61) ITKRORCDHODHSSTR5LCK
SCHEMBL807743 0.87 ITK (0.57) ITKRORCDHODHSSTR5LCK
SCHEMBL807541 0.87 ITK (0.55) ITKRORCDHODHSSTR5TBK1
SCHEMBL10285825 0.85 ITK (0.58) ITKRORCDHODHSSTR5LCK
SCHEMBL807716 0.84 ITK (0.60) ITKRORCDHODHLCKAURKB
SCHEMBL807822 0.84 ITK (0.81) ITKRORCDHODHSSTR5LCK
SCHEMBL808081 0.83 ITK (0.54) ITKRORCDHODHSSTR5TBK1
SCHEMBL2395616 0.82 ITK (0.56) ITKRORCDHODHSSTR5LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035055-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-22 WO disclosed