SCHEMBL807916

SCHEMBL807916

Cc1nccn1Cc1cc(Nc2nc3ccc(Br)cc3s2)nc(N2CCCC(N)C2)c1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 10/20 0.37
PIM2 Q9P1W9 3/20 0.34
MAPT P10636 2/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HTT P42858 1/20 0.34
RAB9A P51151 1/20 0.34
TP53 P04637 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
SYK P43405 1/20 0.34
CXCR3 P49682 1/20 0.34
CYP3A4 P08684 2/20 0.33
PIM1 P11309 2/20 0.33
PIM3 Q86V86 1/20 0.33
MAP4K4 O95819 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2399270 0.83 APP (0.37) MAPTNPC1ALDH1A1HTTRAB9A
SCHEMBL2370319 0.79 LMNA (0.42) MAPTNPC1ALDH1A1RAB9ATP53
SCHEMBL2370368 0.78 ITK (0.47) MAPTNPC1RAB9ATP53RXFP1
SCHEMBL2370365 0.78 ITK (0.47) MAPTNPC1RAB9ATP53RXFP1
SCHEMBL2371227 0.75 APP (0.37) MAPTNPC1ALDH1A1HTTRAB9A
SCHEMBL2371233 0.74 HTT (0.45) MAPTALDH1A1HTTRAB9ARXFP1
SCHEMBL2370208 0.73 ALDH1A1 (0.44) MAPTALDH1A1HTTRXFP1
SCHEMBL807801 0.69 LMNA (0.42) MAPTTP53RXFP1
SCHEMBL2425957 0.67 PIK3CG (0.43)
SCHEMBL2425952 0.67 PIK3CG (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035055-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-22 WO disclosed