SCHEMBL807993

SCHEMBL807993

C=C(/N=C(N)\N=C(/N)c1noc(-c2cccc(F)c2)n1)N(C)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.39
TP53 P04637 2/20 0.38
GPBAR1 Q8TDU6 1/20 0.35
SLC9A1 P19634 1/20 0.35
HDAC1 Q13547 3/20 0.33
HDAC6 Q9UBN7 3/20 0.33
HDAC8 Q9BY41 2/20 0.33
ABCG2 Q9UNQ0 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.32
SCD5 Q86SK9 1/20 0.32
PPARG P37231 2/20 0.32
PPARD Q03181 2/20 0.32
PPARA Q07869 2/20 0.32
S1PR1 P21453 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
NPC1 O15118 1/20 0.32
NFKB1 P19838 1/20 0.32
RAB9A P51151 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10287186 0.87 NPC1 (0.41) GRM5TP53HDAC1NPC1NFKB1
SCHEMBL808333 0.84 NPC1 (0.37) GPBAR1HDAC1HDAC6HDAC8SIGMAR1
SCHEMBL808235 0.82 HDAC6 (0.34) HDAC1HDAC6HDAC8SIGMAR1NPC1
SCHEMBL10287187 0.82 ALDH1A1 (0.45) TP53HDAC1S1PR1NPC1NFKB1
SCHEMBL808234 0.81 HDAC6 (0.34) HDAC1HDAC6HDAC8NPC1RAB9A
SCHEMBL808224 0.80 SIGMAR1 (0.32) SIGMAR1
SCHEMBL808211 0.80 RPS6KA2 (0.33) TP53GPBAR1SIGMAR1NPC1RAB9A
SCHEMBL808221 0.79 SIGMAR1 (0.32) SIGMAR1
SCHEMBL808229 0.79 SIGMAR1 (0.32) SIGMAR1
SCHEMBL807906 0.78 SMN1; SMN2 (0.40) TP53GPBAR1NPC1NFKB1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035023-A1 TRIAZINE-OXADIAZOLES NOVARTIS AG (CH) 2012-03-22 WO disclosed