SCHEMBL808234

SCHEMBL808234

C=C(/N=C(N)\N=C(/N)c1noc(-c2ccc(C(C)=O)nc2)n1)N(C)c1ccccc1

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.34
HDAC1 Q13547 2/20 0.34
HDAC8 Q9BY41 2/20 0.33
HDAC4 P56524 1/20 0.33
KDM1A O60341 1/20 0.31
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10287152 0.94 HDAC6 (0.34) HDAC6HDAC1HDAC8HDAC4KDM1A
SCHEMBL808241 0.88 HDAC6 (0.33) HDAC6HDAC1HDAC8HDAC4
SCHEMBL808236 0.87 TSHR (0.39) HDAC6HDAC1HDAC8KDM1ANPC1
SCHEMBL10287197 0.86 CPT2 (0.33) KDM1ANPC1RAB9A
SCHEMBL10286912 0.85 GABRA1 (0.36) HDAC6HDAC1HDAC8HDAC4
SCHEMBL808237 0.85 HIF1A (0.39)
SCHEMBL808333 0.82 NPC1 (0.37) HDAC6HDAC1HDAC8HDAC4NPC1
SCHEMBL808235 0.81 HDAC6 (0.34) HDAC6HDAC1HDAC8HDAC4NPC1
SCHEMBL10287187 0.81 ALDH1A1 (0.45) HDAC1NPC1RAB9A
SCHEMBL807993 0.81 GRM5 (0.39) HDAC6HDAC1HDAC8HDAC4NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035023-A1 TRIAZINE-OXADIAZOLES NOVARTIS AG (CH) 2012-03-22 WO disclosed