SCHEMBL808235

SCHEMBL808235

C=Cc1ccc(-c2nc(/C(N)=N/C(N)=N\C(=C)N(C)c3ccccc3)no2)cc1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.34
HDAC1 Q13547 2/20 0.34
HDAC8 Q9BY41 2/20 0.33
SIGMAR1 Q99720 1/20 0.32
HDAC4 P56524 1/20 0.31
NPC1 O15118 1/20 0.30
NFKB1 P19838 1/20 0.30
RAB9A P51151 1/20 0.30
NFKB2 Q00653 1/20 0.30
RELA Q04206 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL808333 0.88 NPC1 (0.37) HDAC6HDAC1HDAC8SIGMAR1HDAC4
SCHEMBL807993 0.82 GRM5 (0.39) HDAC6HDAC1HDAC8SIGMAR1HDAC4
SCHEMBL808234 0.81 HDAC6 (0.34) HDAC6HDAC1HDAC8HDAC4NPC1
SCHEMBL808240 0.80 HDAC6 (0.35) HDAC6HDAC1HDAC8HDAC4
SCHEMBL808221 0.79 SIGMAR1 (0.32) SIGMAR1
SCHEMBL808229 0.79 SIGMAR1 (0.32) SIGMAR1
SCHEMBL808224 0.78 SIGMAR1 (0.32) SIGMAR1
SCHEMBL807976 0.78 SIGMAR1 (0.31) SIGMAR1
SCHEMBL807994 0.78 SIGMAR1 (0.31) SIGMAR1
SCHEMBL807937 0.77 GABRA5 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035023-A1 TRIAZINE-OXADIAZOLES NOVARTIS AG (CH) 2012-03-22 WO disclosed