SCHEMBL808042

SCHEMBL808042

C=C(/N=C(N)\N=C(/N)c1noc(-c2ccc(C(F)(F)F)cn2)n1)N(C)c1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LIPE Q05469 3/20 0.35
POLQ O75417 1/20 0.35
CASP3 P42574 2/20 0.33
HDAC4 P56524 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
NPSR1 Q6W5P4 2/20 0.33
STAT3 P40763 2/20 0.33
KDM4E B2RXH2 1/20 0.32
MAPK1 P28482 1/20 0.32
NPC1 O15118 1/20 0.31
S1PR1 P21453 1/20 0.31
S1PR3 Q99500 1/20 0.31
S1PR5 Q9H228 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL807976 0.87 SIGMAR1 (0.31)
SCHEMBL808247 0.85 STAT3 (0.30) STAT3
SCHEMBL10287199 0.82 GABRA5 (0.39) HDAC4HDAC8HDAC6
SCHEMBL10287560 0.80 HDAC4 (0.33) POLQHDAC4HDAC8HDAC6
SCHEMBL808224 0.79 SIGMAR1 (0.32)
SCHEMBL808229 0.78 SIGMAR1 (0.32)
SCHEMBL807993 0.77 GRM5 (0.39) HDAC4HDAC8HDAC6NPC1S1PR1
SCHEMBL808333 0.76 NPC1 (0.37) LIPECASP3HDAC4HDAC8HDAC6
SCHEMBL807994 0.76 SIGMAR1 (0.31)
SCHEMBL10287782 0.76 MAOB (0.36) KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035023-A1 TRIAZINE-OXADIAZOLES NOVARTIS AG (CH) 2012-03-22 WO disclosed