SCHEMBL8080971

SCHEMBL8080971

O=C(OCC1(O)CCCc2ccccc2C1O)N(c1ccccc1)c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGIR P43119 8/20 0.61
PTGDR Q13258 5/20 0.46
PTGER1 P34995 2/20 0.46
PTGER3 P43115 2/20 0.46
CHRM3 P20309 3/20 0.36
CHRM4 P08173 2/20 0.36
CHRM1 P11229 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
CHRM5 P08912 1/20 0.36
CAMK2A Q9UQM7 1/20 0.36
PTGER4 P35408 1/20 0.34
PTGER2 P43116 1/20 0.34
ATM Q13315 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
HTR2A P28223 2/20 0.34
HTR2C P28335 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7717829 0.85 PTGIR (0.65) PTGIRPTGDRPTGER1PTGER3CHRM3
SCHEMBL7718277 0.81 PTGIR (0.89) PTGIRPTGDRPTGER1PTGER3PTGER4
SCHEMBL8078053 0.79 PTGIR (0.43) PTGIRPTGDRPTGER1PTGER3CHRM3
SCHEMBL8082944 0.76 PTGIR (0.63) PTGIRPTGDRPTGER1PTGER3CHRM3
SCHEMBL7779787 0.76 PTGIR (1.00) PTGIRPTGDRPTGER1PTGER3PTGER4
SCHEMBL7720284 0.76 PTGIR (0.61) PTGIRPTGDRPTGER1PTGER3
SCHEMBL8078275 0.74 PTGIR (0.48) PTGIRPTGDRPTGER1PTGER3CHRM3
SCHEMBL7778581 0.72 PTGIR (0.81) PTGIRPTGDRPTGER1PTGER3
SCHEMBL8068504 0.72 BLM (0.54) PTGIRPTGDRPTGER1PTGER3CHRM3
SCHEMBL9017290 0.71 PTGIR (0.44) PTGIRPTGDRPTGER1PTGER3CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1030834-A1 BENZOCYCLOHEPTENE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-08-30 EP disclosed
WO-1999024397-A1 BENZOCYCLOHEPTENE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-05-20 WO disclosed