SCHEMBL8081791

SCHEMBL8081791

CC1=C(C(=O)OC(C)C)C(c2cccc(Cl)c2Cl)C2=C(CCCC2=O)N1C

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PYGL P06737 10/20 0.44
PYGM P11217 10/20 0.44
WDR5 P61964 1/20 0.41
LMNA P02545 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HSD17B10 Q99714 2/20 0.40
TSHR P16473 2/20 0.40
ALOX15 P16050 1/20 0.40
ADORA2B P29275 1/20 0.40
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 2/20 0.39
GAA P10253 2/20 0.39
CASP1 P29466 2/20 0.39
HPGD P15428 1/20 0.39
CASP7 P55210 1/20 0.39
POLB P06746 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8086877 0.89 TSHR (0.45) WDR5LMNAL3MBTL1HSD17B10TSHR
SCHEMBL8080963 0.85 KMT2A (0.47) PYGLPYGMLMNAL3MBTL1TSHR
SCHEMBL7981102 0.80 HSD17B10 (0.64) LMNAHSD17B10TSHRALOX15ALDH1A1
SCHEMBL8086984 0.76 PYGL (0.45) PYGLPYGMLMNAL3MBTL1ALOX15
SCHEMBL10653191 0.72 PYGL (0.53) PYGLPYGMLMNAHSD17B10TSHR
SCHEMBL7275567 0.72 PYGL (0.49) PYGLPYGMLMNAHSD17B10TSHR
SCHEMBL9046285 0.72 KMT2A (0.45) PYGLPYGMLMNAL3MBTL1TSHR
SCHEMBL8086890 0.71 NPSR1 (0.65) WDR5LMNAHSD17B10TSHRALDH1A1
SCHEMBL9048171 0.70 HSD17B10 (0.49) HSD17B10TSHRALOX15ALDH1A1KDM4E
SCHEMBL7979577 0.69 KDM4E (0.62) HSD17B10TSHRALOX15ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6121284-A SPECIFIED 1-(ALKYL OR CYCLOALKYL)-2-METHYL-3-(ALKOXYCARBONYL)-4-(SUBSTITUTED PYRIDYL OR ARYL)-5-OXO-1,4,5,6,7,8-HEXAHYDROQUINOLINE COMPOUNDS; TREATING SICKLE CELL ANEMIA, PSYCHOSES, DEPRESSION BAYER AKTIENGESELLSCHAFT (DE) 2000-09-19 US claimed