SCHEMBL8086984

SCHEMBL8086984

CC1=C(C(=O)OC(C)C)C(c2cccc(Cl)c2Cl)C2=C(C(=O)OC2)N1C

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PYGL P06737 14/20 0.45
PYGM P11217 14/20 0.45
LMNA P02545 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ADORA2B P29275 2/20 0.41
ALOX15 P16050 1/20 0.41
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
POLB P06746 1/20 0.39
HTT P42858 1/20 0.39
ALOX12 P18054 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9045340 0.86 PYGL (0.36) PYGLPYGMLMNAL3MBTL1ADORA2B
SCHEMBL8082470 0.79 ALOX15 (0.51) PYGLPYGMLMNAL3MBTL1ADORA2B
SCHEMBL8081791 0.76 PYGL (0.44) PYGLPYGMLMNAL3MBTL1ADORA2B
SCHEMBL8080963 0.74 KMT2A (0.47) PYGLPYGMLMNAL3MBTL1ADORA2B
SCHEMBL10653191 0.73 PYGL (0.53) PYGLPYGMLMNAALOX15ALDH1A1
SCHEMBL7275567 0.72 PYGL (0.49) PYGLPYGMLMNAALDH1A1
SCHEMBL9047294 0.69 ALOX15 (0.40) PYGLPYGMLMNAL3MBTL1ALOX15
SCHEMBL9770221 0.69 PYGM (0.52) PYGLPYGMLMNAL3MBTL1ALDH1A1
SCHEMBL9658365 0.69 PYGL (0.42) PYGLPYGMLMNAALOX15ALDH1A1
SCHEMBL8080875 0.69 ADORA2B (0.41) PYGLPYGMLMNAADORA2BALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6121284-A SPECIFIED 1-(ALKYL OR CYCLOALKYL)-2-METHYL-3-(ALKOXYCARBONYL)-4-(SUBSTITUTED PYRIDYL OR ARYL)-5-OXO-1,4,5,6,7,8-HEXAHYDROQUINOLINE COMPOUNDS; TREATING SICKLE CELL ANEMIA, PSYCHOSES, DEPRESSION BAYER AKTIENGESELLSCHAFT (DE) 2000-09-19 US disclosed