SCHEMBL808244

SCHEMBL808244

C=C(/N=C(N)\N=C(/N)c1noc(-c2ccc(COCC(F)(F)F)nc2)n1)Nc1ccccc1

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 12/20 0.34
HDAC1 Q13547 10/20 0.34
HDAC8 Q9BY41 9/20 0.34
SCN9A Q15858 2/20 0.33
HDAC5 Q9UQL6 5/20 0.33
KCNH2 Q12809 1/20 0.32
SCN5A Q14524 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10287127 0.87 HDAC8 (0.33) HDAC6HDAC1HDAC8HDAC5
SCHEMBL10287133 0.86 CNR2 (0.31)
SCHEMBL808249 0.85 HDAC4 (0.30) HDAC1
SCHEMBL10287198 0.84 HDAC6 (0.34) HDAC6HDAC1HDAC8SCN9AHDAC5
SCHEMBL10287123 0.76 POLB (0.41) HDAC6HDAC1HDAC8SCN9A
SCHEMBL808041 0.74 TRPV1 (0.39)
SCHEMBL808240 0.72 HDAC6 (0.35) HDAC6HDAC1HDAC8HDAC5
SCHEMBL10287296 0.72 ATR (0.42)
SCHEMBL10287533 0.71 ADRA2A (0.33)
SCHEMBL795333 0.70 PIK3CA (0.41) HDAC6HDAC1HDAC8SCN9AHDAC5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035023-A1 TRIAZINE-OXADIAZOLES NOVARTIS AG (CH) 2012-03-22 WO disclosed