SCHEMBL808041

SCHEMBL808041

C=C(/N=C(N)\N=C(/N)c1noc(-c2ncccc2C(F)(F)F)n1)Nc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 14/20 0.39
ADRA2A P08913 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA2C P18825 1/20 0.31
ATR Q13535 1/20 0.31
GAA P10253 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10287533 0.88 ADRA2A (0.33) ADRA2AADRA2BADRA2C
SCHEMBL10287560 0.82 HDAC4 (0.33) TRPV1
SCHEMBL808249 0.75 HDAC4 (0.30)
SCHEMBL808244 0.74 HDAC6 (0.34)
SCHEMBL10287136 0.67 ALDH1A1 (0.41) GAA
SCHEMBL795790 0.66 AURKA (0.41) TRPV1GAA
SCHEMBL10287123 0.65 POLB (0.41)
SCHEMBL808315 0.64 SMN1; SMN2 (0.39)
SCHEMBL807957 0.63 LMNA (0.41) GAA
SCHEMBL807959 0.61 NPSR1 (0.33) ADRA2AADRA2BADRA2CGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035023-A1 TRIAZINE-OXADIAZOLES NOVARTIS AG (CH) 2012-03-22 WO disclosed