SCHEMBL10287296

SCHEMBL10287296

C=C(/N=C(N)\N=C(/N)c1noc(-c2ccnc(OC)c2)n1)Nc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.42
S1PR1 P21453 3/20 0.41
CNR1 P21554 1/20 0.37
USP30 Q70CQ3 1/20 0.35
HAVCR2 Q8TDQ0 5/20 0.34
ALOX5AP P20292 1/20 0.34
KDM4E B2RXH2 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
TP53 P04637 2/20 0.33
MAPT P10636 2/20 0.33
MEN1 O00255 1/20 0.33
TSHR P16473 1/20 0.33
XBP1 P17861 1/20 0.33
PPARG P37231 1/20 0.33
KMT2A Q03164 1/20 0.33
NCOA2 Q15596 1/20 0.33
HSD17B10 Q99714 1/20 0.33
POLB P06746 1/20 0.33
WNT3A P56704 1/20 0.33
BUB1 O43683 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10287533 0.76 ADRA2A (0.33) ALDH1A1
SCHEMBL10287136 0.73 ALDH1A1 (0.41) S1PR1KDM4ESMN1; SMN2TP53MAPT
SCHEMBL808244 0.72 HDAC6 (0.34)
SCHEMBL10287123 0.69 POLB (0.41) HAVCR2TP53MAPTMEN1KMT2A
SCHEMBL808249 0.69 HDAC4 (0.30)
SCHEMBL15477231 0.66 S1PR1 (0.50) ATRS1PR1USP30ALOX5APKDM4E
SCHEMBL10287187 0.66 ALDH1A1 (0.45) S1PR1KDM4ESMN1; SMN2TP53MAPT
SCHEMBL24921187 0.64 S1PR1 (0.64) S1PR1USP30ALOX5APKDM4ESMN1; SMN2
SCHEMBL807993 0.64 GRM5 (0.39) S1PR1SMN1; SMN2TP53MAPTPPARG
SCHEMBL808315 0.64 SMN1; SMN2 (0.39) SMN1; SMN2MEN1TSHRKMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035023-A1 TRIAZINE-OXADIAZOLES NOVARTIS AG (CH) 2012-03-22 WO disclosed