SCHEMBL8083017

SCHEMBL8083017

CNC1CC=CC2CN(c3c(F)cc4c(=O)c(C(=O)O)cn(C5CC5F)c4c3Cl)CC21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.49
POLB P06746 3/20 0.49
OPRM1 P35372 2/20 0.49
CHRM2 P08172 1/20 0.49
CHRM1 P11229 1/20 0.49
OPRD1 P41143 1/20 0.49
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
LMNA P02545 2/20 0.37
KDM4E B2RXH2 6/20 0.37
HPGD P15428 5/20 0.37
HSD17B10 Q99714 4/20 0.37
ALB P02768 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
KCNH2 Q12809 5/20 0.37
TOP1 P11387 1/20 0.37
AADAT Q8N5Z0 2/20 0.36
TUBB4A P04350 1/20 0.36
TUBB P07437 1/20 0.36
TUBA3C P0DPH7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8091231 0.93 KDM4E (0.40) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL8083224 0.91 ALDH1A1 (0.59) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9047303 0.90 ALDH1A1 (0.39) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL8089691 0.83 TOP2A (0.49) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9047385 0.83 KDM4E (0.32) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL8091409 0.82 KDM4E (0.40) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9044116 0.81 ALDH1A1 (0.47) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL8092759 0.80 ALDH1A1 (0.54) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9053933 0.79 ALDH1A1 (0.59) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9053930 0.79 ALDH1A1 (0.59) ALDH1A1POLBOPRM1CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6018054-A INTERMEDIATE COMPOUNDS FOR PREPARING NOVEL QUINOLONE AND NAPHTHYRIDONE DERIVATIVES WHICH ARE SUBSTITUTED IN THE 7-POSITION BY A PARTIALLY HYDROGENATED ISOINDOLINYL RING, USE AS ANTIBACTERIAL AGENTS AND AS FEED ADDITIVES BAYER AKTIENGESELLSCHAFT (DE) 2000-01-25 US disclosed
US-5556979-A ANIMAL FEEDS BAYER AKTIENGESELLSCHAFT (DE) 1996-09-17 US disclosed