SCHEMBL8083373

SCHEMBL8083373

CCOC(=O)c1ccc(CCc2ccc3cccnc3n2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SUCNR1 Q9BXA5 5/20 0.45
MAOB P27338 1/20 0.45
NPC1 O15118 4/20 0.45
RAB9A P51151 4/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
MAPT P10636 3/20 0.44
LMNA P02545 1/20 0.44
NAMPT P43490 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
HPGD P15428 1/20 0.43
CYP2C19 P33261 1/20 0.43
PTPN1 P18031 1/20 0.42
NFKB1 P19838 1/20 0.42
MAPK1 P28482 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20024878 0.78 SUCNR1 (0.46) SUCNR1MAPTLMNAHPGDALDH1A1
SCHEMBL6743269 0.78 LMNA (0.50) NPC1RAB9ASMN1; SMN2LMNANAMPT
SCHEMBL20139157 0.78 MAOB (0.45) SUCNR1MAOBNPC1RAB9ASMN1; SMN2
SCHEMBL12199135 0.77 CA1 (0.68) NPC1RAB9ASMN1; SMN2MAPTLMNA
SCHEMBL7562110 0.76 ALDH1A1 (0.47) MAOBNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL7562106 0.76 ALDH1A1 (0.47) MAOBNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL14237207 0.76 KDM4E (0.59) MAOBMAPTLMNACYP1A2HPGD
SCHEMBL6265814 0.76 SUCNR1 (0.53) SUCNR1HPGDALDH1A1TP53
SCHEMBL5260948 0.76 NPC1 (0.53) NPC1RAB9ASMN1; SMN2MAPTLMNA
SCHEMBL21281662 0.76 MAOB (0.44) SUCNR1MAOBSMN1; SMN2MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6017925-A Integrin antagonists MERCK & CO., INC. (US) 2000-01-25 US disclosed
US-5929120-A Guainidino, formamidino, amino and related compounds for inhibiting osteoclast-mediated bone resorption MERCK & CO., INC. (US) 1999-07-27 US disclosed
US-5741796-A Pyridyl and naphthyridyl compounds for inhibiting osteoclast-mediated bone resorption MERCK & CO., INC. (US) 1998-04-21 US disclosed
EP-0760658-A4 COMPOUNDS FOR INHIBITING OSTEOCLAST-MEDIATED BONE RESORPTION MERCK & CO INC (US) 1997-09-17 EP disclosed
EP-0760658-A1 COMPOUNDS FOR INHIBITING OSTEOCLAST-MEDIATED BONE RESORPTION MERCK & CO. INC. (US) 1997-03-12 EP disclosed
WO-1995032710-A1 COMPOUNDS FOR INHIBITING OSTEOCLAST-MEDIATED BONE RESORPTION MERCK & CO., INC. (US) 1995-12-07 WO disclosed