SCHEMBL8083391

SCHEMBL8083391

[CH2]c1cccc(N(CC(C)C)S(=O)(=O)c2cccc3nc(N)sc23)c1O

nearest known ligand 0.32

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RORC P51449 3/20 0.32
KMT2A Q03164 1/20 0.32
MCL1 Q07820 2/20 0.31
HSD11B1 P28845 1/20 0.31
NR1H4 Q96RI1 1/20 0.30
TSHR P16473 1/20 0.30
BCL2L1 Q07817 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7450471 0.81 RORC (0.39) RORCKMT2AMCL1BCL2L1
SCHEMBL5174385 0.81 ALDH1A1 (0.45) RORCKMT2AMCL1BCL2L1
SCHEMBL7609854 0.75 RORC (0.39) RORCKMT2AMCL1BCL2L1
SCHEMBL7343868 0.74 RORC (0.47) RORCMCL1BCL2L1
SCHEMBL2578313 0.73 MCL1 (0.50) RORCMCL1BCL2L1
SCHEMBL7451743 0.73 RORC (0.45) RORCMCL1TSHRBCL2L1
SCHEMBL7450627 0.72 RORC (0.46) RORCMCL1BCL2L1
SCHEMBL5031155 0.69 RORC (0.40) RORC
SCHEMBL2576483 0.69 SPPL2A (0.35) RORC
SCHEMBL7452491 0.68 KEAP1 (0.50) RORCMCL1BCL2L1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE43802-E1 α- and β-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors G.D. SEARLE LLC (US) 2012-11-13 US claimed
US-6140505-A REACTING A BENZO FUSED HETEROCYCLIC COMPOUND WITH AN SO3 COMPLEX IN THE PRESENCE OF A WATER IMMISCIBLE, NON-REACTIVE SOLVENT, AT A TEMPERATURE OF FROM ABOUT 0 TO ABOUT 75 DEGREES C., COOLING AND THEN ADDING OXALYL HALIDE. G. D. SEARLE & CO. (US) 2000-10-31 US disclosed