SCHEMBL8083552

SCHEMBL8083552

NCCCC[CH]NC(=O)c1ccc(C23CCC(Cl)(CC2)CC3)cc1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSB P07858 1/20 0.33
CYP1A2 P05177 1/20 0.31
TSHR P16473 1/20 0.31
NFKB1 P19838 1/20 0.31
MAOB P27338 1/20 0.31
MEN1 O00255 1/20 0.31
BLM P54132 1/20 0.31
PMP22 Q01453 1/20 0.31
KMT2A Q03164 1/20 0.31
SMYD3 Q9H7B4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8091498 0.96 CYP1A2 (0.32) CYP1A2TSHRNFKB1MAOBMEN1
SCHEMBL8095262 0.85 HDAC3 (0.32) CYP1A2TSHRNFKB1MAOB
SCHEMBL8095325 0.85 POLB (0.33) CTSB
SCHEMBL8095242 0.84 SPHK1 (0.32)
SCHEMBL8091503 0.81 SMYD3 (0.47) CYP1A2TSHRNFKB1MAOBMEN1
SCHEMBL8091664 0.81 POLB (0.33)
SCHEMBL8083555 0.80 NAMPT (0.46) CYP1A2TSHRNFKB1MAOBMEN1
SCHEMBL8091492 0.73 CTSB (0.38) CTSB
SCHEMBL8090161 0.72 SPHK1 (0.33)
SCHEMBL8083595 0.71 CTSB (0.34) CTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0792883-B1 Novel derivates of boronic acid, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 2000-12-20 EP disclosed
EP-0792883-A1 Novel derivates of boronic acid, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1997-09-03 EP disclosed