SCHEMBL8083976

SCHEMBL8083976

Nc1cc(C2(S(=O)(=O)c3ccc(Cl)cc3)CC2)nc(-c2ccc(NC(=O)Nc3ccccn3)cc2)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.52
RAB9A P51151 3/20 0.52
MEN1 O00255 5/20 0.43
KMT2A Q03164 5/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
CNR1 P21554 3/20 0.43
KDM4E B2RXH2 1/20 0.41
MAPT P10636 1/20 0.41
ADORA3 P0DMS8 1/20 0.40
PIM1 P11309 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA2B P29275 1/20 0.40
ADORA1 P30542 1/20 0.40
FLT3 P36888 1/20 0.40
PIM3 Q86V86 1/20 0.40
AURKB Q96GD4 1/20 0.40
SMARCA2 P51531 1/20 0.40
SMARCA4 P51532 1/20 0.40
MTOR P42345 4/20 0.40
PIK3CA P42336 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8083683 0.92 NPC1 (0.42) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL8092270 0.88 NPC1 (0.43) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL8091838 0.85 KMT2A (0.43) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL8099638 0.84 FLT3 (0.43) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL8084738 0.82 PIK3CA (0.40) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL8098775 0.82 CA1 (0.43) MEN1KMT2ACNR1KDM4EMAPT
SCHEMBL8098814 0.81 EPHX1 (0.47) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL3925969 0.81 PIK3CA (0.51) MTORPIK3CAPIK3R1PIK3CG
SCHEMBL8096186 0.81 MAPT (0.41) KDM4EMAPTPIK3CAKDRLMNA
SCHEMBL8092289 0.81 CA1 (0.41) CNR1KDM4EMAPTMTORPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed