SCHEMBL8092270

SCHEMBL8092270

Nc1cc(C2(S(=O)(=O)c3ccccn3)CC2)nc(-c2ccc(NC(=O)Nc3ccccn3)cc2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.43
RAB9A P51151 7/20 0.43
FLT3 P36888 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
ADORA3 P0DMS8 1/20 0.43
PIM1 P11309 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA2B P29275 1/20 0.43
ADORA1 P30542 1/20 0.43
PIM3 Q86V86 1/20 0.43
AURKB Q96GD4 1/20 0.43
LMNA P02545 3/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
KDM4E B2RXH2 1/20 0.40
PIK3CA P42336 4/20 0.40
MTOR P42345 4/20 0.40
LIMK1 P53667 1/20 0.39
PIK3R1 P27986 2/20 0.39
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8096070 0.90 MTOR (0.40) KMT2APIK3CAMTORPIK3R1ATR
SCHEMBL8093540 0.90 RAB9A (0.39) NPC1RAB9AFLT3MEN1KMT2A
SCHEMBL8096681 0.89 ATR (0.40) MEN1KMT2AKDM4EPIK3CAMTOR
SCHEMBL8083683 0.88 NPC1 (0.42) NPC1RAB9AFLT3SMN1; SMN2ADORA3
SCHEMBL8083976 0.88 NPC1 (0.52) NPC1RAB9AFLT3SMN1; SMN2ADORA3
SCHEMBL8092294 0.88 ROCK2 (0.39) NPC1PIK3CAMTORLIMK1PIK3R1
SCHEMBL8098135 0.87 MTOR (0.39) PIK3CAMTORPIK3R1ATR
SCHEMBL8099638 0.87 FLT3 (0.43) NPC1RAB9AFLT3SMN1; SMN2ADORA3
SCHEMBL8091129 0.86 KDR (0.40) RAB9AFLT3SMN1; SMN2ATRKIT
SCHEMBL8091924 0.86 NAMPT (0.39) RAB9APIK3CAATRKITKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed