SCHEMBL8083683

SCHEMBL8083683

Nc1cc(C2(S(=O)(=O)c3ccc(F)cc3)CC2)nc(-c2ccc(NC(=O)Nc3ccccn3)cc2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 8/20 0.42
RAB9A P51151 8/20 0.42
LMNA P02545 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.40
ADORA3 P0DMS8 1/20 0.40
PIM1 P11309 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA2B P29275 1/20 0.40
ADORA1 P30542 1/20 0.40
FLT3 P36888 1/20 0.40
PIM3 Q86V86 1/20 0.40
AURKB Q96GD4 1/20 0.40
PIK3CA P42336 5/20 0.40
MTOR P42345 5/20 0.40
PIK3R1 P27986 2/20 0.40
PIK3CG P48736 1/20 0.38
KMT2A Q03164 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8083976 0.92 NPC1 (0.52) NPC1RAB9ALMNACYP1A2CYP2C9
SCHEMBL8092270 0.88 NPC1 (0.43) NPC1RAB9ALMNACYP1A2CYP2C9
SCHEMBL8083973 0.85 ALDH1A1 (0.43) NPC1RAB9APIK3CAMTORPIK3R1
SCHEMBL8083200 0.84 ALDH1A1 (0.43) PIK3CAMTORPIK3R1PIK3CGKMT2A
SCHEMBL8099638 0.84 FLT3 (0.43) NPC1RAB9ALMNACYP1A2CYP2C9
SCHEMBL8098812 0.83 NPC1 (0.43) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL8084738 0.82 PIK3CA (0.40) NPC1RAB9ALMNASMN1; SMN2ADORA3
SCHEMBL8099408 0.81 CA2 (0.42) PIK3CAMTORKMT2AMEN1CA12
SCHEMBL8097689 0.81 ALDH1A1 (0.40) LMNAPIK3CAMTORPIK3R1PIK3CG
SCHEMBL8092946 0.81 ABL1 (0.41) NPC1RAB9ASMN1; SMN2PIK3CAPIK3R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed