SCHEMBL8084522

SCHEMBL8084522

CCc1ccccc1NCCCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.51
GAA P10253 1/20 0.51
KMT2A Q03164 3/20 0.50
SIGMAR1 Q99720 3/20 0.50
MEN1 O00255 2/20 0.50
GRM2 Q14416 1/20 0.50
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
HPGD P15428 1/20 0.49
POLB P06746 1/20 0.49
HDAC1 Q13547 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
KDM6B O15054 1/20 0.48
KDM4C Q9H3R0 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8093196 0.95 L3MBTL1 (0.53) HDAC6GAAKMT2ASIGMAR1MEN1
SCHEMBL6513356 0.89 GAA (0.54) GAAKMT2ASIGMAR1MEN1GRM2
SCHEMBL3966040 0.82 POLB (0.60) HDAC6GAACYP2C9CYP2C19POLB
SCHEMBL30806170 0.81 MAPT (0.54) HDAC6GAAKMT2ASIGMAR1MEN1
SCHEMBL10407866 0.80 POLB (0.54) HDAC6GAASIGMAR1CYP2C9CYP2C19
SCHEMBL18289061 0.80 ALDH1A1 (0.43) GAAHPGDPOLBL3MBTL1
SCHEMBL19495506 0.79 HSD17B10 (0.53) GAAGRM2HPGDPOLBHDAC8
Hydrochloric Acid SCHEMBL2343034 0.79 MAPT (0.52) HDAC6GAAKMT2ASIGMAR1MEN1
SCHEMBL11598417 0.79 MAPT (0.64) HDAC6GAAKMT2ASIGMAR1MEN1
SCHEMBL10407954 0.79 POLB (0.53) POLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057371-A TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS, GASTROINTESTINAL DISORDERS, DRUG ABUSE, ANGINA, MIGRAINE, HYPERTENSION AND DEPRESSION VIRGINIA COMMONWEALTH UNIVERSITY (US) 2000-05-02 US disclosed
EP-0591426-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1994-04-13 EP disclosed
WO-1993000313-A2 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1993-01-07 WO disclosed